Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 6568
TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139465BDBM139465(US8889672, 317-080-001)
Affinity DataIC50: 1.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139466BDBM139466(US8889672, 317-094-001)
Affinity DataIC50: 2.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139467BDBM139467(US8889672, 268-020-002)
Affinity DataIC50: 2.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139483BDBM139483(US8889672, 194-094-003)
Affinity DataIC50: 3.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139468BDBM139468(US8889672, 317-054-001)
Affinity DataIC50: 4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139480BDBM139480(US8889672, 194-074-005)
Affinity DataIC50: 4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139481BDBM139481(US8889672, 194-074-008)
Affinity DataIC50: 4.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139484BDBM139484(US8889672, 194-094-009)
Affinity DataIC50: 5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139469BDBM139469(US8889672, 317-052-004)
Affinity DataIC50: 5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139482BDBM139482(US8889672, 194-094-008)
Affinity DataIC50: 5.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139470BDBM139470(US8889672, 317-056-002)
Affinity DataIC50: 6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139471BDBM139471(US8889672, 317-120-001)
Affinity DataIC50: 6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139464BDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50: 6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139472BDBM139472(US8889672, 252-036-001)
Affinity DataIC50: 6.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139473BDBM139473(US8889672, 227-076-001)
Affinity DataIC50: 7.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139474BDBM139474(US8889672, 317-052-001)
Affinity DataIC50: 7.00E+3nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139475BDBM139475(US8889672, 268-044-002)
Affinity DataIC50: 1.10E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139478BDBM139478(US8889672, 317-048-002)
Affinity DataIC50: 1.70E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139464BDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50: 2.00E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139477BDBM139477(US8889672, 317-008-004)
Affinity DataIC50: 2.00E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139476BDBM139476(US8889672, 317-010-004)
Affinity DataIC50: 2.10E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139488BDBM139488(US8889672, 5632675 | US8889672, 5627112)
Affinity DataIC50: 2.40E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139486BDBM139486(US8889672, 5132573)
Affinity DataIC50: 2.60E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139488BDBM139488(US8889672, 5632675 | US8889672, 5627112)
Affinity DataIC50: 2.80E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139464BDBM139464(US8889672, 194-074-007 | US8889672, PKCzI-diMeO)
Affinity DataIC50: 3.50E+4nMAssay Description:IC50 values were determined using an in vitro luminescence-based kinase assay against aPKCζ to elucidate a pharmacophore. The IC50 values determ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139489BDBM139489(US8889672, APOGEE A)
Affinity DataIC50: 3.90E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139487BDBM139487(US8889672, 5311310)
Affinity DataIC50: 4.10E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139491BDBM139491(US8889672, 5635527)
Affinity DataIC50: 6.20E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent

TargetProtein kinase C zeta type(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 139492BDBM139492(US8889672, APOGEE B)
Affinity DataIC50: 7.10E+4nMAssay Description:The IC50 values for PKCl-diMeO and compounds described herein and illustrated in FIG. 6 are described in Table 2. The IC50 values were determined usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/27/2015
Entry Details
US Patent