Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 6651
TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143179BDBM143179(US9266895, 4 | US8940744, 4)
Affinity DataIC50: 0.300nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143181BDBM143181(US9266895, 6 | US8940744, 6)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143191BDBM143191(US9266895, 13 | US8940744, 13 | US11040980, Exampl...)
Affinity DataIC50: 0.600nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143203BDBM143203(US9266895, 22 | US8940744, 22 | US9994576, 22 | US...)
Affinity DataIC50: 0.600nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143202BDBM143202(US9266895, 21 | US8940744, 21 | US9994576, 21 | US...)
Affinity DataIC50: 0.700nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143198BDBM143198(US9266895, 18 | US8940744, 18 | US9994576, 18 | US...)
Affinity DataIC50: 0.700nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143192BDBM143192(US9266895, 13a | US8940744, 13a | US9994576, 13a |...)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143182BDBM143182(US9266895, 7 | US8940744, 7 | US9994576, 7 | US110...)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143217BDBM143217(US9266895, 8A | US8940744, 8A | US9994576, 8A)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143201BDBM143201(US9266895, 20 | US8940744, 20 | US9994576, 20 | US...)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143204BDBM143204(US9266895, 23 | US8940744, 23 | US9994576, 23 | US...)
Affinity DataIC50: 1nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143205BDBM143205(US9266895, 24 | US8940744, 24 | US9994576, 24 | US...)
Affinity DataIC50: 1.20nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143215BDBM143215(US9266895, 34 | US8940744, 34 | US9994576, 34 | US...)
Affinity DataIC50: 1.30nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143206BDBM143206(US9266895, 25 | US8940744, 25 | US9994576, 25 | US...)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143212BDBM143212(US9266895, 31 | US8940744, 31 | US9994576, 31 | US...)
Affinity DataIC50: 1.5nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143199BDBM143199(US9266895, 19 | US8940744, 19 | US9994576, 19 | US...)
Affinity DataIC50: 1.5nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143213BDBM143213(US9266895, 32 | US8940744, 32 | US9994576, 32 | US...)
Affinity DataIC50: 1.90nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143180BDBM143180(US9266895, 5 | US8940744, 5 | US9994576, 5 | US110...)
Affinity DataIC50: 1.90nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143214BDBM143214(US9266895, 33 | US8940744, 33 | US9994576, 33 | US...)
Affinity DataIC50: 2nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143185BDBM143185(US9266895, 10 | US8940744, 10 | US9994576, 10 | US...)
Affinity DataIC50: 2.10nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143176BDBM143176(US9266895, 1 | US8940744, 1 | US9994576, 1 | US110...)
Affinity DataIC50: 3.10nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143183BDBM143183(US9266895, 8 | US8940744, 8 | US9994576, 8 | US110...)
Affinity DataIC50: 3.80nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143190BDBM143190(US9266895, 12 | US8940744, 12 | US9994576, 12 | US...)
Affinity DataIC50: 4nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143177BDBM143177(US9266895, 2 | US8940744, 2 | US9994576, 2)
Affinity DataIC50: 4.10nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143195BDBM143195(US9266895, 15 | US8940744, 15 | US9994576, 15 | US...)
Affinity DataIC50: 4.10nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143184BDBM143184(US9266895, 9 | US8940744, 9 | US9994576, 9 | US110...)
Affinity DataIC50: 4.70nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143211BDBM143211(US9266895, 30 | US8940744, 30 | US9994576, 30 | US...)
Affinity DataIC50: 5.20nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143200BDBM143200(US8940744, 19a)
Affinity DataIC50: 5.60nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143178BDBM143178(US9266895, 3 | US8940744, 3 | US9994576, 3)
Affinity DataIC50: 8.10nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143216BDBM143216(US9266895, 35 | US8940744, 35 | US9994576, 35 | US...)
Affinity DataIC50: 13nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143188BDBM143188(US9266895, 11 | US8940744, 11 | US9994576, 11 | US...)
Affinity DataIC50: 16.1nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143194BDBM143194(US9266895, 14 | US8940744, 14 | US9994576, 14 | US...)
Affinity DataIC50: 20.4nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143193BDBM143193(US9266895, 13b | US8940744, 13b | US9994576, 13b |...)
Affinity DataIC50: 26nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent