Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 7353
TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190690BDBM190690(US9181233, 67)
Affinity DataKi:  10nM ΔG°:  -46.4kJ/mole IC50: 80nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190685BDBM190685(US9181233, 60)
Affinity DataKi:  40nM ΔG°:  -42.9kJ/mole IC50: 450nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190679BDBM190679(US9181233, 52)
Affinity DataKi:  50nM ΔG°:  -42.4kJ/mole IC50: 680nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190680BDBM190680(US9181233, 54)
Affinity DataKi:  60nM ΔG°:  -41.9kJ/mole IC50: 590nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190676BDBM190676(US9181233, 47)
Affinity DataKi:  60nM ΔG°:  -41.9kJ/mole IC50: 400nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190678BDBM190678(US9181233, 50)
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 760nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190695BDBM190695(US9181233, 86)
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 290nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190671BDBM190671(US9181233, 10)
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 480nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190687BDBM190687(US9181233, 62)
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 480nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190681BDBM190681(US9181233, 55)
Affinity DataKi:  80nM ΔG°:  -41.2kJ/mole IC50: 490nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190677BDBM190677(US9181233, 49)
Affinity DataKi:  90nM ΔG°:  -40.9kJ/mole IC50: 360nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190694BDBM190694(US9181233, 85)
Affinity DataKi:  100nM ΔG°:  -40.6kJ/mole IC50: 470nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190688BDBM190688(US9181233, 63)
Affinity DataKi:  100nM ΔG°:  -40.6kJ/mole IC50: 220nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190669BDBM190669(US9181233, 8)
Affinity DataKi:  110nM ΔG°:  -40.4kJ/mole IC50: 640nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190693BDBM190693(US9181233, 84)
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 570nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190696BDBM190696(US9181233, 87)
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 550nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190689BDBM190689(US9181233, 65)
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 530nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190672BDBM190672(US9181233, 22)
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 520nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190684BDBM190684(US9181233, 59)
Affinity DataKi:  120nM ΔG°:  -40.2kJ/mole IC50: 560nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190674BDBM190674(US9181233, 39)
Affinity DataKi:  130nM ΔG°:  -40.0kJ/mole IC50: 800nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190682BDBM190682(US9181233, 57)
Affinity DataKi:  130nM ΔG°:  -40.0kJ/mole IC50: 830nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190692BDBM190692(US9181233, 83)
Affinity DataKi:  140nM ΔG°:  -39.8kJ/mole IC50: 570nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190683BDBM190683(US9181233, 58)
Affinity DataKi:  140nM ΔG°:  -39.8kJ/mole IC50: 720nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190691BDBM190691(US9181233, 68)
Affinity DataKi:  150nM ΔG°:  -39.6kJ/mole IC50: 410nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190686BDBM190686(US9181233, 61)
Affinity DataKi:  170nM ΔG°:  -39.3kJ/mole IC50: 760nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190675BDBM190675(US9181233, 46)
Affinity DataKi:  180nM ΔG°:  -39.1kJ/mole IC50: 640nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190670BDBM190670(US9181233, 9)
Affinity DataKi:  200nM ΔG°:  -38.9kJ/mole IC50: 760nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase-like protein(Human)
Probiodrug

US Patent
LigandChemical structure of BindingDB Monomer ID 190673BDBM190673(US9181233, 24)
Affinity DataKi:  230nM ΔG°:  -38.5kJ/mole IC50: 850nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2016
Entry Details
US Patent