Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 407 Enz. Inhib. hit(s) with all data for entry = 7829
TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM144940(US8952157, 122 | US9303025, 122)
Affinity DataKi: <0.00100nM ΔG°: <-68.5kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145154(US8952157, 345 | US9303025, 345)
Affinity DataKi:  0.00500nM ΔG°:  -64.5kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM144855(US8952157, 37 | US9303025, 37)
Affinity DataKi:  0.00500nM ΔG°:  -64.5kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145152(US8952157, 343 | US9303025, 343)
Affinity DataKi:  0.00900nM ΔG°:  -63.0kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145179(US8952157, 370 | US9303025, 370)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145180(US8952157, 371 | US9303025, 371)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145099(US8952157, 289 | US9303025, 289)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145022(US8952157, 209 | US9303025, 209)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145014(US8952157, 201 | US9303025, 201)
Affinity DataKi:  0.0100nM ΔG°:  -62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145011(US8952157, 198 | US9303025, 198)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145177(US8952157, 368 | US9303025, 368)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145172(US8952157, 363 | US9303025, 363)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145159(US8952157, 350 | US9303025, 350)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145155(US8952157, 346 | US9303025, 346)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145147(US8952157, 338 | US9303025, 338)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145145(US8952157, 336 | US9303025, 336)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145144(US8952157, 335 | US9303025, 335)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145139(US8952157, 330 | US9303025, 330)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145133(US8952157, 324 | US9303025, 324)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145127(US8952157, 318 | US9303025, 318)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145122(US8952157, 313 | US9303025, 313)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145187(US8952157, 378 | US9303025, 378)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145194(US8952157, 385 | US9303025, 386)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145196(US8952157, 387 | US9303025, 387)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145198(US8952157, 389 | US9303025, 389)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145199(US8952157, 390 | US9303025, 390)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145200(US8952157, 391 | US9303025, 391)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145201(US8952157, 392 | US9303025, 392)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145202(US8952157, 393 | US9303025, 393)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145205(US8952157, 396 | US9303025, 396)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145208(US8952157, 399 | US9303025, 399)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145219(US8952157, 410 | US9303025, 410)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145106(US8952157, 296 | US9303025, 296)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM221452(US9303025, 297)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145111(US8952157, 302 | US9303025, 302)
Affinity DataKi: <0.0100nM ΔG°: <-62.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145176(US8952157, 367 | US9303025, 367)
Affinity DataKi:  0.0120nM ΔG°:  -62.3kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM144970(US8952157, 154 | US9303025, 154)
Affinity DataKi:  0.0120nM ΔG°:  -62.3kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM144856(US8952157, 38 | US9303025, 38)
Affinity DataKi:  0.0130nM ΔG°:  -62.1kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145173(US8952157, 364 | US9303025, 364)
Affinity DataKi:  0.0140nM ΔG°:  -62.0kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145178(US8952157, 369 | US9303025, 369)
Affinity DataKi:  0.0140nM ΔG°:  -62.0kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145170(US8952157, 361 | US9303025, 361)
Affinity DataKi:  0.0150nM ΔG°:  -61.8kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145162(US8952157, 353 | US9303025, 353)
Affinity DataKi:  0.0160nM ΔG°:  -61.6kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM221448(US9303025, 138)
Affinity DataKi:  0.0160nM ΔG°:  -61.6kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145150(US8952157, 341 | US9303025, 341)
Affinity DataKi:  0.0170nM ΔG°:  -61.5kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145098(US8952157, 288 | US9303025, 288)
Affinity DataKi:  0.0170nM ΔG°:  -61.5kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145087(US8952157, 277 | US9303025, 277)
Affinity DataKi:  0.0170nM ΔG°:  -61.5kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145203(US8952157, 394 | US9303025, 394)
Affinity DataKi:  0.0180nM ΔG°:  -61.3kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM145158(US8952157, 349 | US9303025, 349)
Affinity DataKi:  0.0190nM ΔG°:  -61.2kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM144858(US8952157, 40 | US9303025, 40)
Affinity DataKi:  0.0190nM ΔG°:  -61.2kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetApoptosis regulator Bcl-2(Human)
Abbvie

US Patent
LigandPNGBDBM144857(US8952157, 39 | US9303025, 39)
Affinity DataKi:  0.0190nM ΔG°:  -61.2kJ/moleT: 25°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 μM (2× starting concentration; 10% DMSO) and 10 μ...More data for this Ligand-Target Pair
In DepthDetails US Patent


Displayed 1 to 50 (of 407 total ) | Next | Last >>
Jump to: