Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 3214
TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394274(US9975902, Example 4)
Affinity DataIC50: 1.00E+4nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394270(US9975902, Example 1)
Affinity DataIC50: 1.00E+4nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394272(US9975902, Example 2)
Affinity DataIC50: 1.00E+4nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394272(US9975902, Example 2)
Affinity DataIC50: 1.00E+4nMAssay Description:The peptidyl-proline isomerase activity (PPase) was determined by using a PPase-chymotrypsin coupled assay with suc-AAPF-p-NA as substrated and color...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394273(US9975902, Example 3)
Affinity DataIC50: 1.00E+4nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394274(US9975902, Example 4)
Affinity DataIC50: 1.05E+5nMAssay Description:The peptidyl-proline isomerase activity (PPase) was determined by using a PPase-chymotrypsin coupled assay with suc-AAPF-p-NA as substrated and color...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394275(US9975902, Example 5)
Affinity DataIC50: 1.05E+5nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394276(US9975902, Example 6)
Affinity DataIC50: 1.05E+5nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394281(US9975902, Example 11)
Affinity DataIC50: 1.05E+5nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394277(US9975902, Example 7)
Affinity DataIC50: 1.05E+5nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394278(US9975902, Example 8)
Affinity DataIC50: 1.05E+5nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394279(US9975902, Example 9)
Affinity DataIC50: 1.05E+5nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase D(Human)
Merck Patent

US Patent
LigandPNGBDBM394280(US9975902, Example 10)
Affinity DataIC50: 1.05E+5nMAssay Description:The binding capacity of the compounds was measured using a competition Fluorescence-Polarisation based assay with fluorescine labelled cyclosporin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent