Compile Data Set for Download or QSAR
Report error Found 123 Enz. Inhib. hit(s) with all data for entry = 3216
LigandPNGBDBM394319(US9975907, Example 39)
Affinity DataIC50: 1nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394323(US9975907, Example 43)
Affinity DataIC50: 1nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394330(US9975907, Example 50 | US10428087, Example 50 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394332(US9975907, Example 52 | US10428087, Example 52 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394292(US9975907, Example 11 | US10428087, Example 11 | U...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394326(US9975907, Example 46 | US10428087, Example 46 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394329(US9975907, Example 49 | US10428087, Example 49 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394289(US9975907, Example 8 | US10428087, Example 8 | US1...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394290(US9975907, Example 9 | US10428087, Example 9 | US1...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394290(US9975907, Example 9 | US10428087, Example 9 | US1...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394325(US9975907, Example 45 | US10428087, Example 45 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394346(US9975907, Example 66 | US10428087, Example 66 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM50004547(CHEMBL2216863 | US9708333, 28 | US10065963, Compou...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394347(US9975907, Example 67 | US10428087, Example 67 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM50004547(CHEMBL2216863 | US9708333, 28 | US10065963, Compou...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394344(US9975907, Example 64 | US10428087, Example 64 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394345(US9975907, Example 65 | US10428087, Example 65 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394338(US9975907, Example 58 | US10428087, Example 58 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394293(US9975907, Example 12 | US9975907, Example 44 | US...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394339(US9975907, Example 59 | US10428087, Example 59 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394294(US9975907, Example 13 | US9975907, Example 23 | US...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394340(US9975907, Example 60 | US10428087, Example 60 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394294(US9975907, Example 13 | US9975907, Example 23 | US...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394292(US9975907, Example 11 | US10428087, Example 11 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394334(US9975907, Example 54 | US10428087, Example 54 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394337(US9975907, Example 57 | US10428087, Example 57 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394294(US9975907, Example 13 | US9975907, Example 23 | US...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394358(US9975907, Example 78 | US10428087, Example 78 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394353(US9975907, Example 73 | US10428087, Example 73 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394300(US9975907, Example 20 | US10428087, Example 20 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394354(US9975907, Example 74 | 2-{1-[(2-Amino-9H-purin-6-...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394301(US9975907, Example 21 | US10428087, Example 21 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM124076(US8754089, 3-(3-fluorophenyl)-6-methyl-2-((1R)-1-(...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394320(US9975907, Example 40 | US10428087, Example 40 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394314(US9975907, Example 34 | US10428087, Example 34 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394283(US9975907, Example 2 | US10428087, Example 2 | US1...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394313(US9975907, Example 33 | US10428087, Example 33 | U...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:PI3-Kinase luminescent assay kit including lipid kinase substrate, D-myo-phosphatidylinositol 4,5-bisphosphate (PtdIns(4,5)P2)D (+)-sn-1,2-di-O-octan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM246889(7-(1-(9H-purin-6- ylamino)ethyl)-6-(3- fluoropheny...)
Affinity DataIC50: 50nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394364(US9975907, Example 84 | US10428087, Example 84aRes...)
Affinity DataIC50: 75nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394357(US9975907, Example 77 | US10428087, Example 77 | U...)
Affinity DataIC50: 75nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394290(US9975907, Example 9 | US10428087, Example 9 | US1...)
Affinity DataIC50: 75nMAssay Description:Materials: Lipid kinase substrate, phosphoinositol-4,5-bisphosphate (PIP2), was purchased from Echelon Biosciences (Salt Lake City, Utah). PI3K isofo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394328(US9975907, Example 48 | US10428087, Example 48 | U...)
Affinity DataIC50: 75nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM394302(US9975907, Example 22 | US10428087, Example 22 | U...)
Affinity DataIC50: 75nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

LigandPNGBDBM124079(US8754089, 3-(3-fluorophenyl)-6-methyl-2-(1-(9H-pu...)
Affinity DataIC50: 75nMAssay Description:The kinase reaction was conducted in polystyrene 384-well matrix white plate from Thermo Fisher Scientific in a final volume of 25 μL. Inhibitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
US Patent

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