Reaction Details Report a problem with these data
Target
Adenosine receptor A1 Isoform 2
Ligand
BDBM601697
Substrate
n/a
Meas. Tech.
Radioligand Binding Assay
Ki
>10000±n/a nM
Citation
Kristensen, JL; Jensen, AA; Märcher-Rørsted, E; Leth-Petersen, S 5-HT2A agonists for use in treatment of depression US Patent US11642336 Publication Date 5/9/2023
More Info.:
Target
Name:
Adenosine receptor A1 Isoform 2
Synonyms:
AA1R_HUMAN | ADORA1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
13352.59
Organism:
Homo sapiens (Human)
Description:
P30542-2
Residue:
125
Sequence:
MPPSISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGALVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRRISQCMASTKS