Reaction Details Report a problem with these data
Target
5-hydroxytryptamine receptor 5A
Ligand
BDBM50288778
Substrate
n/a
Meas. Tech.
ChEBML_1530
Ki
58±n/a nM
Citation
Appelberg, U; Mohell, N; Hacksell, U Derivatives of 2-arylcyclopropylamine: Synthesis and interactions with 5-HT1A receptors. Bioorg Med Chem Lett 6:415-420 (1996) Article
More Info.:
Target
Name:
5-hydroxytryptamine receptor 5A
Synonyms:
5-HT-5A | 5-HT5a | 5-hydroxytryptamine receptor 5A | 5HT5A_RAT | 5ht5a | Htr5a | REC17 | Serotonin (5-HT) receptor | Serotonin receptor 5A
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40684.21
Organism:
RAT
Description:
5-HT5a HTR5A RAT::P35364
Residue:
357
Sequence:
MDLPINLTSFSLSTPSTLEPNRSLDTEALRTSQSFLSAFRVLVLTLLGFLAAATFTWNLLVLATILRVRTFHRVPHNLVASMAISDVLVAVLVMPLSLVHELSGRRWQLGRRLCQLWIACDVLCCTASIWNVTAIALDRYWSITRHLEYTLRARKRVSNVMILLTWALSAVISLAPLLFGWGETYSELSEECQVSREPSYTVFSTVGAFYLPLCVVLFVYWKIYKAAKFRMGSRKTNSVSPIPEAVEVKDASQHPQMVFTVRHATVTFQTEGDTWREQKEQRAALMVGILIGVFVLCWFPFFVTELISPLCSWDIPALWKSIFLWLGYSNSFFNPLIYTAFNRSYSSAFKVFFSKQQ