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Target
PAS domain-containing serine/threonine-protein kinase [879-1323]
Ligand
BDBM487229
Substrate
n/a
Meas. Tech.
Radiochemical Assay
IC50
<10000±n/a nM
Citation
McCall, JM; Kelly, RC; Romero, DL Heterocyclic compounds for the inhibition of pask US Patent US10953012 Publication Date 3/23/2021
More Info.:
Target
Name:
PAS domain-containing serine/threonine-protein kinase [879-1323]
Synonyms:
KIAA0135 | PAS domain-containing serine/threonine-protein kinase (PASK) (879-1323) | PASK | PASK_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49711.83
Organism:
Homo sapiens (Human)
Description:
aa 879-1323
Residue:
445
Sequence:
MRGAAGLQREIQEGAYSGSCYHRDGLRLSIQFEVRRVELQGPTPLFCCWLVKDLLHSQRDSAARTRLFLASLPGSTHSTAAELTGPSLVEVLRARPWFEEPPKAVELEGLAACEGEYSQKYSTMSPLGSGAFGFVWTAVDKEKNKEVVVKFIKKEKVLEDCWIEDPKLGKVTLEIAILSRVEHANIIKVLDIFENQGFFQLVMEKHGSGLDLFAFIDRHPRLDEPLASYIFRQLVSAVGYLRLKDIIHRDIKDENIVIAEDFTIKLIDFGSAAYLERGKLFYTFCGTIEYCAPEVLMGNPYRGPELEMWSLGVTLYTLVFEENPFCELEETVEAAIHPPYLVSKELMSLVSGLLQPVPERRTTLEKLVTDPWVTQPVNLADYTWEEVFRVNKPESGVLSAASLEMGNRSLSDVAQAQELCGGPVPGEAPNGQGCLHPGDPRLLTS