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Target
Sliding-clamp-loader large/small subunit
Ligand
BDBM36319
Substrate
BDBM50118233
Meas. Tech.
colorimetric ATPase assay
pH
7.5±0
Temperature
298.15±0 K
Ki
4.8e+3± 5e+2 nM
Citation
More Info.:
Target
Name:
Sliding-clamp-loader large/small subunit
Synonyms:
ATP-dependent clamp loaders gp44/62
Type:
n/a
Mol. Mass.:
n/a
Description:
n/a
Components:
This complex has 2 components.
Component 1
Name:
Sliding-clamp-loader large subunit
Synonyms:
44 | Clamp loader large subunit | Gene product 44 | LOADL_BPT4 | Sliding-clamp-loader gp44 subunit | gp44
Type:
n/a
Mol. Mass.:
35788.87
Organism:
Enterobacteria phage T4
Description:
P04526
Residue:
319
Sequence:
MITVNEKEHILEQKYRPSTIDECILPAFDKETFKSITSKGKIPHIILHSPSPGTGKTTVAKALCHDVNADMMFVNGSDCKIDFVRGPLTNFASAASFDGRQKVIVIDEFDRSGLAESQRHLRSFMEAYSSNCSIIITANNIDGIIKPLQSRCRVITFGQPTDEDKIEMMKQMIRRLTEICKHEGIAIADMKVVAALVKKNFPDFRKTIGELDSYSSKGVLDAGILSLVTNDRGAIDDVLESLKNKDVKQLRALAPKYAADYSWFVGKLAEEIYSRVTPQSIIRMYEIVGENNQYHGIAANTELHLAYLFIQLACEMQWK
Component 2
Name:
Sliding-clamp-loader small subunit
Synonyms:
62 | Clamp loader small subunit | Gene product 62 | LOADS_BPT4 | Sliding-clamp-loader gp44 subunit | gp62
Type:
n/a
Mol. Mass.:
21366.49
Organism:
Enterobacteria phage T4
Description:
P04527
Residue:
187
Sequence:
MSLFKDDIQLNEHQVAWYSKDWTAVQSAADSFKEKAENEFFEIIGAINNKTKCSIAQKDYSKFMVENALSQFPECMPAVYAMNLIGSGLSDEAHFNYLMAAVPRGKRYGKWAKLVEDSTEVLIIKLLAKRYQVNTNDAINYKSILTKNGKLPLVLKELKGLVTDDFLKEVTKNVKEQKQLKKLALEW
Inhibitor
Name:
BDBM36319
Synonyms:
5-nitro-indolyl- 2'-deoxyriboside triphosphate | d5-NITP
Type:
Small organic molecule
Emp. Form.:
C13H17N2O14P3
Mol. Mass.:
518.2004
SMILES:
[H][C@]1(O)C[C@@]([H])(O[C@]1([H])COP(O)(=O)OP(O)(=O)OP(O)(O)=O)n1ccc2cc(ccc12)[N+]([O-])=O