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Target
Somatostatin receptor type 5
Ligand
BDBM50468132
Substrate
n/a
Meas. Tech.
ChEMBL_1798124 (CHEMBL4270241)
IC50
7.4±n/a nM
Citation
Liu, W; Shao, PP; Liang, GB; Bawiec, J; He, J; Aster, SD; Wu, M; Chicchi, G; Wang, J; Tsao, KL; Shang, J; Salituro, G; Zhou, YP; Li, C; Akiyama, TE; Metzger, DE; Murphy, BA; Howard, AD; Weber, AE; Duffy, JL Discovery and Pharmacology of a Novel Somatostatin Subtype 5 (SSTR5) Antagonist: Synergy with DPP-4 Inhibition. ACS Med Chem Lett 9:1082-1087 (2018) [PubMed] Article
More Info.:
Target
Name:
Somatostatin receptor type 5
Synonyms:
SS-5-R | SS5-R | SS5R | SSR5_MOUSE | Smstr5 | Somatostatin receptor | Somatostatin receptor 5 | Somatostatin receptor type 5 | Sstr5
Type:
PROTEIN
Mol. Mass.:
40022.97
Organism:
Mus musculus
Description:
ChEMBL_833921
Residue:
362
Sequence:
MEPLSLTSTPSWNASAASSSSHNWSLVDPVSPMGARAVLVPVLYLLVCTVGLGGNTLVIYVVLRYAKMKTVTNVYILNLAVADVLFMLGLPFLATQNAVSYWPFGSFLCRLVMTLDGINQFTSIFCLMVMSVDRYLAVVHPLRSARWRRPRVAKLASAAVWVFSLLMSLPLLVFADVQEGWGTCNLSWPEPVGLWGAAFITYTSVLGFFGPLLVICLCYLLIVVKVKAAGMRVGSSRRRRSERKVTRMVVVVVLVFVGCWLPFFIVNIVNLAFTLPEEPTSAGLYFFVVVLSYANSCANPLLYGFLSDNFRQSFRKALCLRRGYGVEDADAIEPRPDKSGRPQTTLPTRSCEANGLMQTSRL