Reaction Details Report a problem with these data
Target
Neuropeptides B/W receptor type 1
Ligand
BDBM50362421
Substrate
n/a
Meas. Tech.
ChEMBL_797950 (CHEMBL1942827)
IC50
16±n/a nM
Citation
Anthony Romero, F; Hastings, NB; Moningka, R; Guo, Z; Wang, M; Di Salvo, J; Lei, Y; Trusca, D; Deng, Q; Tong, V; Terebetski, JL; Ball, RG; Ujjainwalla, F The discovery of potent antagonists of NPBWR1 (GPR7). Bioorg Med Chem Lett 22:1014-8 (2012) [PubMed] Article
More Info.:
Target
Name:
Neuropeptides B/W receptor type 1
Synonyms:
G-protein coupled receptor 7 | Gpr7 | NPBW1_MOUSE | Npbwr1
Type:
PROTEIN
Mol. Mass.:
36085.77
Organism:
Mouse
Description:
ChEMBL_797950
Residue:
329
Sequence:
MHNLTLFESGGDNVSCGGSSLGCPNGSSLAPLPLPQPLAVAVPVVYGVICAVGLAGNSAVLYVLLRTPRMKTVTNVFILNLAIADELFTLVLPINIADFLLRRWPFGEVMCKLIVAVDQYNTFSSLYFLAVMSADRYLVVLATAESRRVSGRTYGAARAVSLAVWALVTLVVLPFAVFARLDEEQGRRQCVLVFPQPEAFWWRASRLYTLVLGFAIPVTTICALYTTLLCRLRAIQLDSHAKALDRAKKRVTLLVAAILAVCLLCWTPYHLSTIVALTTDLPQTPLVIGISYFITSLSYANSCLNPFLYAFLDDSFRRSLRQLVSCRSA