Reaction Details Report a problem with these data
Target
Galanin peptides
Ligand
BDBM85190
Substrate
n/a
Ki
2600±n/a nM
Comments
PDSP_1276
Citation
Johansson, L; Sohn, D; Thorberg, SO; Jackson, DM; Kelder, D; Larsson, LG; Rényi, L; Ross, SB; Wallsten, C; Eriksson, H; Hu, PS; Jerning, E; Mohell, N; Westlind-Danielsson, A The pharmacological characterization of a novel selective 5-hydroxytryptamine1A receptor antagonist, NAD-299. J Pharmacol Exp Ther 283:216-25 (1997) [PubMed]
More Info.:
Target
Name:
Galanin peptides
Synonyms:
GALANIN | GALA_RAT | Gal | Galanin peptides | Galn
Type:
Enzyme Catalytic Domain
Mol. Mass.:
13327.23
Organism:
Rat
Description:
GALANIN 0 RAT::P10683
Residue:
124
Sequence:
MARGSVILLAWLLLVATLSATLGLGMPTKEKRGWTLNSAGYLLGPHAIDNHRSFSDKHGLTGKRELPLEVEEGRLGSVAVPLPESNIVRTIMEFLSFLHLKEAGALDSLPGIPLATSSEDLEQS