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Target
L-lactate dehydrogenase
Ligand
BDBM93299
Substrate
n/a
Meas. Tech.
Enzyme Assay
IC50
4.3e+4±n/a nM
Citation
Choi, SR; Beeler, AB; Pradhan, A; Watkins, EB; Rimoldi, JM; Tekwani, B; Avery, MA Generation of oxamic acid libraries: antimalarials and inhibitors of Plasmodium falciparum lactate dehydrogenase. J Comb Chem 9:292-300 (2007) [PubMed] Article
More Info.:
Target
Name:
L-lactate dehydrogenase
Synonyms:
Lactate dehydrogenase (LDH)
Type:
Protein
Mol. Mass.:
28939.78
Organism:
Plasmodium falciparum
Description:
B9UDZ5
Residue:
267
Sequence:
LIVKKNLGDVVLFDIVKNMPHGKALDTSHTNVMAYSNCKVSGSNTYDDLAGADVVIVTAGFTKAPGKSDKEWNRDDLLPLNNKIMIEIGGHIKKNCPNAFIIVVTNPVDVMVQLLHQHSGVPKNKIIGLGGVLDTSRLKYYISQKLNVCPRDVNAHIVGAHGNKMVLLKRYITVGGIPLQEFINNKLISDAELEAIFDRTVNTALEIVNLHASPYVAPAAAIIEMAESYLKDLKKVLICSTLLEGQYGHSDIFGGTPVVLGANGVEQ