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Target
DNA-directed RNA polymerase subunit alpha
Ligand
BDBM466522
Substrate
n/a
Meas. Tech.
Assay of Inhibition of Escherichia coli RNA Polymerase
IC50
530±n/a nM
Citation
Ebright, RH; Shen, J Arylpropionyl-triketone antibacterial agents US Patent US10800725 Publication Date 10/13/2020
More Info.:
Target
Name:
DNA-directed RNA polymerase subunit alpha
Synonyms:
JW3257 | RNA polymerase subunit alpha | RNAP subunit alpha | RPOA_ECOLI | Transcriptase subunit alpha | pez | phs | rpoA | sez
Type:
PROTEIN
Mol. Mass.:
36497.18
Organism:
Escherichia coli K-12
Description:
ChEMBL_106172
Residue:
329
Sequence:
MQGSVTEFLKPRLVDIEQVSSTHAKVTLEPLERGFGHTLGNALRRILLSSMPGCAVTEVEIDGVLHEYSTKEGVQEDILEILLNLKGLAVRVQGKDEVILTLNKSGIGPVTAADITHDGDVEIVKPQHVICHLTDENASISMRIKVQRGRGYVPASTRIHSEEDERPIGRLLVDACYSPVERIAYNVEAARVEQRTDLDKLVIEMETNGTIDPEEAIRRAATILAEQLEAFVDLRDVRQPEVKEEKPEFDPILLRPVDDLELTVRSANCLKAEAIHYIGDLVQRTEVELLKTPNLGKKSLTEIKDVLASRGLSLGMRLENWPPASIADE