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Target
C-C motif chemokine 3
Ligand
BDBM65497
Substrate
n/a
Meas. Tech.
cytomteric bead array (CBA) assay
Temperature
310.15±n/a K
IC50
28±n/a nM
Comments
extracted
Citation
 Gandhi, A; Dimartino, J; Chopra, R Methods for the treatment of locally advanced breast cancer US Patent  US9694015 Publication Date 7/4/2017 
Target
Name:
C-C motif chemokine 3
Synonyms:
CCL3 | CCL3_HUMAN | G0/G1 switch regulatory protein 19-1 | G0S19-1 | MIP-1-alpha | MIP1A | Macrophage inflammatory protein 1-alpha | PAT 464.1 | SCYA3 | SIS-beta | Small-inducible cytokine A3 | Tonsillar lymphocyte LD78 alpha protein
Type:
Protein
Mol. Mass.:
10083.38
Organism:
Homo sapiens (Human)
Description:
P10147
Residue:
92
Sequence:
MQVSTAALAVLLCTMALCNQFSASLAADTPTACCFSYTSRQIPQNFIADYFETSSQCSKPGVIFLTKRSRQVCADPSEEWVQKYVSDLELSA
  
Inhibitor
Name:
BDBM65497
Synonyms:
CC-220 (Compound 6) | US9694015, 6.4S
Type:
Small organic molecule
Emp. Form.:
C25H27N3O5
Mol. Mass.:
449.499
SMILES:
O=C1N(Cc2c1cccc2OCc1ccc(CN2CCOCC2)cc1)[C@H]1CCC(=O)NC1=O
Structure:
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