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Target
Tyrosine-protein phosphatase YopH
Ligand
BDBM34775
Substrate
n/a
Meas. Tech.
YopH - IC50 determinations (10 point dose range)
IC50
46893.19229±n/a nM
Citation
 PubChem, PC YopH - IC50 determinations (10 point dose range) PubChem Bioassay (2008)[AID] 
Target
Name:
Tyrosine-protein phosphatase YopH
Synonyms:
YOPH_YEREN | yop51 | yopH
Type:
PROTEIN
Mol. Mass.:
50951.99
Organism:
Yersinia enterocolitica
Description:
ChEMBL_965525
Residue:
468
Sequence:
MNLSLSDLHRQVSRLVQQESGDCTGKLRGNVAANKETTFQGLTIASGARESEKVFAQTVLSHVANIVLTQEDTAKLLQSTVKHNLNNYELRSVGNGNSVLVSLRSDQMTLQDAKVLLEAALRQESGARGHVSSHSHSVLHAPGTPVREGLRSHLDPRTPPLPPRERPHTSGHHGAGEARATAPSTVSPYGPEARAELSSRLTTLRNTLAPATNDPRYLQACGGEKLNRFRDIQCCRQTAVRADLNANYIQVGNTRTIACQYPLQSQLESHFRMLAENRTPVLAVLASSSEIANQRFGMPDYFRQSGTYGSITVESKMTQQVGLGDGIMADMYTLTIREAGQKTISVPVVHVGNWPDQTAVSSEVTKALASLVDQTAETKRNMYESKGSSAVADDSKLRPVIHCRAGVGRTAQLIGAMCMNDSRNSQLSVEDMVSQMRVQRNGIMVQKDEQLDVLIKLAEGQGRPLLNS
  
Inhibitor
Name:
BDBM34775
Synonyms:
1-Ethyl-2,3-dimethyl-2-phenyl-2,3-dihydro-1H-benzoimidazole | 1-ethyl-2,3-dimethyl-2-phenyl-benzimidazole | 1-ethyl-2,3-dimethyl-2-phenylbenzimidazole | MLS000567447 | SMR000176391 | cid_3124417
Type:
Small organic molecule
Emp. Form.:
C17H20N2
Mol. Mass.:
252.3541
SMILES:
CCN1c2ccccc2N(C)C1(C)c1ccccc1
Structure:
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