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Target
Sialidase-1
Ligand
BDBM50270454
Substrate
n/a
Meas. Tech.
ChEMBL_1789505 (CHEMBL4261239)
Ki
830±n/a nM
Citation
Guo, T; Héon-Roberts, R; Zou, C; Zheng, R; Pshezhetsky, AV; Cairo, CW Selective Inhibitors of Human Neuraminidase 1 (NEU1). J Med Chem 61:11261-11279 (2018) [PubMed] Article
More Info.:
Target
Name:
Sialidase-1
Synonyms:
NANH | NEU1 | NEUR1_HUMAN | Sialidase 1
Type:
PROTEIN
Mol. Mass.:
45463.28
Organism:
Homo sapiens (Human)
Description:
ChEMBL_960639
Residue:
415
Sequence:
MTGERPSTALPDRRWGPRILGFWGGCRVWVFAAIFLLLSLAASWSKAENDFGLVQPLVTMEQLLWVSGRQIGSVDTFRIPLITATPRGTLLAFAEARKMSSSDEGAKFIALRRSMDQGSTWSPTAFIVNDGDVPDGLNLGAVVSDVETGVVFLFYSLCAHKAGCQVASTMLVWSKDDGVSWSTPRNLSLDIGTEVFAPGPGSGIQKQREPRKGRLIVCGHGTLERDGVFCLLSDDHGASWRYGSGVSGIPYGQPKQENDFNPDECQPYELPDGSVVINARNQNNYHCHCRIVLRSYDACDTLRPRDVTFDPELVDPVVAAGAVVTSSGIVFFSNPAHPEFRVNLTLRWSFSNGTSWRKETVQLWPGPSGYSSLATLEGSMDGEEQAPQLYVLYEKGRNHYTESISVAKISVYGTL