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Target
Serine/threonine-protein kinase 16
Ligand
BDBM50273541
Substrate
n/a
Meas. Tech.
ChEMBL_1806405 (CHEMBL4305764)
Ki
11900±n/a nM
Citation
Verdonck, S; Pu, SY; Sorrell, FJ; Elkins, JM; Froeyen, M; Gao, LJ; Prugar, LI; Dorosky, DE; Brannan, JM; Barouch-Bentov, R; Knapp, S; Dye, JM; Herdewijn, P; Einav, S; De Jonghe, S Synthesis and Structure-Activity Relationships of 3,5-Disubstituted-pyrrolo[2,3- b]pyridines as Inhibitors of Adaptor-Associated Kinase 1 with Antiviral Activity. J Med Chem 62:5810-5831 (2019) [PubMed] Article
More Info.:
Target
Name:
Serine/threonine-protein kinase 16
Synonyms:
MPSK1 | PKL12 | STK16 | STK16_HUMAN | Serine/threonine-protein kinase 16 | TSF1 | Tyrosine-protein kinase STK16 (STK16)
Type:
Protein
Mol. Mass.:
34659.07
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
305
Sequence:
MGHALCVCSRGTVIIDNKRYLFIQKLGEGGFSYVDLVEGLHDGHFYALKRILCHEQQDREEAQREADMHRLFNHPNILRLVAYCLRERGAKHEAWLLLPFFKRGTLWNEIERLKDKGNFLTEDQILWLLLGICRGLEAIHAKGYAHRDLKPTNILLGDEGQPVLMDLGSMNQACIHVEGSRQALTLQDWAAQRCTISYRAPELFSVQSHCVIDERTDVWSLGCVLYAMMFGEGPYDMVFQKGDSVALAVQNQLSIPQSPRHSSALRQLLNSMMTVDPHQRPHIPLLLSQLEALQPPAPGQHTTQI