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Target
Proteasome subunit beta type-4
Ligand
BDBM50185646
Substrate
n/a
Meas. Tech.
ChEMBL_361597 (CHEMBL859725)
Ki
>80000±n/a nM
Citation
Basse, N; Papapostolou, D; Pagano, M; Reboud-Ravaux, M; Bernard, E; Felten, AS; Vanderesse, R Development of lipopeptides for inhibiting 20S proteasomes. Bioorg Med Chem Lett 16:3277-81 (2006) [PubMed] Article
More Info.:
Target
Name:
Proteasome subunit beta type-4
Synonyms:
PRE1 | PSB4_YEAST | Proteasome Macropain subunit
Type:
PROTEIN
Mol. Mass.:
22515.40
Organism:
Saccharomyces cerevisiae
Description:
ChEMBL_361597
Residue:
198
Sequence:
MDIILGIRVQDSVILASSKAVTRGISVLKDSDDKTRQLSPHTLMSFAGEAGDTVQFAEYIQANIQLYSIREDYELSPQAVSSFVRQELAKSIRSRRPYQVNVLIGGYDKKKNKPELYQIDYLGTKVELPYGAHGYSGFYTFSLLDHHYRPDMTTEEGLDLLKLCVQELEKRMPMDFKGVIVKIVDKDGIRQVDDFQAQ