Reaction Details Report a problem with these data
Target
Platelet-derived growth factor subunit A
Ligand
BDBM99471
Substrate
n/a
Meas. Tech.
ChEMBL_1296291 (CHEMBL3132619)
IC50
610±n/a nM
Citation
Okaniwa, M; Hirose, M; Arita, T; Yabuki, M; Nakamura, A; Takagi, T; Kawamoto, T; Uchiyama, N; Sumita, A; Tsutsumi, S; Tottori, T; Inui, Y; Sang, BC; Yano, J; Aertgeerts, K; Yoshida, S; Ishikawa, T Discovery of a selective kinase inhibitor (TAK-632) targeting pan-RAF inhibition: design, synthesis, and biological evaluation of C-7-substituted 1,3-benzothiazole derivatives. J Med Chem 56:6478-94 (2013) [PubMed] Article
More Info.:
Target
Name:
Platelet-derived growth factor subunit A
Synonyms:
PDGF subunit A | PDGF-1 | PDGF1 | PDGFA | PDGFA_HUMAN | Platelet-derived growth factor A chain | Platelet-derived growth factor alpha polypeptide
Type:
PROTEIN
Mol. Mass.:
24060.81
Organism:
Homo sapiens (Human)
Description:
ChEMBL_108150
Residue:
211
Sequence:
MRTLACLLLLGCGYLAHVLAEEAEIPREVIERLARSQIHSIRDLQRLLEIDSVGSEDSLDTSLRAHGVHATKHVPEKRPLPIRRKRSIEEAVPAVCKTRTVIYEIPRSQVDPTSANFLIWPPCVEVKRCTGCCNTSSVKCQPSRVHHRSVKVAKVEYVRKKPKLKEVQVRLEEHLECACATTSLNPDYREEDTGRPRESGKKRKRKRLKPT