Reaction Details Report a problem with these data
Target
Apamin
Ligand
BDBM50049750
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_218
Citation
Sullivan, JP; Donnelly-Roberts, D; Briggs, CA; Anderson, DJ; Gopalakrishnan, M; Piattoni-Kaplan, M; Campbell, JE; McKenna, DG; Molinari, E; Hettinger, AM; Garvey, DS; Wasicak, JT; Holladay, MW; Williams, M; Arneric, SP A-85380 [3-(2(S)-azetidinylmethoxy) pyridine]: in vitro pharmacological properties of a novel, high affinity alpha 4 beta 2 nicotinic acetylcholine receptor ligand. Neuropharmacology 35:725-34 (1996) [PubMed] Article
More Info.:
Target
Name:
Apamin
Synonyms:
APAM_APIME | Apamine
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5226.87
Organism:
Apis mellifera (Honeybee)
Description:
Potassium channel, Apamin 0 0::P01500
Residue:
46
Sequence:
MISMLRCIYLFLSVILITSYFVTPVMPCNCKAPETALCARRCQQHG