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Found 351 with Last Name = 'garvey' and Initial = 'ds'
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081496(5-((S)-1-Azetidin-2-ylmethoxy)-pyrimidine | CHEMBL...)
Affinity DataKi:  0.130nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049756(3-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyridine |...)
Affinity DataKi:  0.150nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081490(5-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyrimidine...)
Affinity DataKi:  2.40nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081484(3-((S)-1-Methyl-pyrrolidin-3-yloxy)-pyridine | CHE...)
Affinity DataKi:  2.70nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50035398((S)-1-Methyl-2-(3-methyl-isoxazol-5-yl)-pyrrolidin...)
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287851((S)-2-(3-Fluoro-phenoxymethyl)-azetidine | CHEMBL3...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081483(3-((R)-1-Methyl-pyrrolidin-3-yloxy)-pyridine | CHE...)
Affinity DataKi:  4.40nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287814((S)-2-(3-Fluoro-phenoxymethyl)-1-methyl-pyrrolidin...)
Affinity DataKi:  5nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAcetylcholine receptor subunit alpha(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  5.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081487(5-((S)-1-Methyl-azetidin-2-ylmethoxy)-pyrimidine |...)
Affinity DataKi:  6.5nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081473(5-(1-Methyl-pyrrolidin-3-yloxy)-pyrimidine | CHEMB...)
Affinity DataKi:  12nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287829((R)-2-(3-Fluoro-phenoxymethyl)-pyrrolidine | CHEMB...)
Affinity DataKi:  13nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287821((S)-2-(3-Fluoro-phenoxymethyl)-1-methyl-azetidine ...)
Affinity DataKi:  14nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287812((S)-2-(3-Fluoro-phenoxymethyl)-pyrrolidine | CHEMB...)
Affinity DataKi:  14nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081476(3-((S)-1-Azetidin-2-ylmethoxy)-6-chloro-pyridazine...)
Affinity DataKi:  15nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081475(2-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyrazine |...)
Affinity DataKi:  16nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287838((S)-2-(3,4-Difluoro-phenoxymethyl)-pyrrolidine | C...)
Affinity DataKi:  17nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287848((S)-2-(3,4-Difluoro-phenoxymethyl)-1-methyl-pyrrol...)
Affinity DataKi:  18nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287816((S)-2-(3,5-Difluoro-phenoxymethyl)-pyrrolidine | C...)
Affinity DataKi:  18nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287834(3-((S)-1-Pyrrolidin-2-ylmethoxy)-benzonitrile | CH...)
Affinity DataKi:  18nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287849((S)-2-(3,5-Difluoro-phenoxymethyl)-1-methyl-pyrrol...)
Affinity DataKi:  19nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005854(1-(4-Azetidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | ...)
Affinity DataKi:  27nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081478(3-((S)-1-Methyl-azetidin-2-ylmethoxy)-pyridazine |...)
Affinity DataKi:  28nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081497(3-Chloro-6-((S)-1-methyl-pyrrolidin-2-ylmethoxy)-p...)
Affinity DataKi:  29nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287852((S)-2-(3-Chloro-phenoxymethyl)-1-methyl-pyrrolidin...)
Affinity DataKi:  37nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081479(3-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-pyridazine...)
Affinity DataKi:  42nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287824((S)-1-Methyl-2-phenoxymethyl-pyrrolidine | CHEMBL7...)
Affinity DataKi:  42nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNicotinic acetylcholine receptor(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50035406(3-Methyl-5-((R)-1-methyl-pyrrolidin-2-yl)-isoxazol...)
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081477(3-Chloro-6-(1-methyl-pyrrolidin-3-yloxy)-pyridazin...)
Affinity DataKi:  46nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287820(3-((S)-1-Methyl-pyrrolidin-2-ylmethoxy)-benzonitri...)
Affinity DataKi:  51nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287843((S)-2-Phenoxymethyl-azetidine | CHEMBL72031)
Affinity DataKi:  52nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081474(3-Chloro-6-((S)-1-methyl-azetidin-2-ylmethoxy)-pyr...)
Affinity DataKi:  64nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287825((S)-2-(2,3-Difluoro-phenoxymethyl)-1-methyl-pyrrol...)
Affinity DataKi:  69nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287846((S)-2-(2,3-Difluoro-phenoxymethyl)-pyrrolidine | C...)
Affinity DataKi:  77nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuronal acetylcholine receptor subunit alpha-10(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287854((R)-2-(3-Fluoro-phenoxymethyl)-1-methyl-pyrrolidin...)
Affinity DataKi:  78nMAssay Description:Binding affinity against neuronal nicotinic acetylcholine receptor(nAChR) by using [3H]-Cytisine as radioligand in whole rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataKi:  84nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50081481(3-Chloro-6-((R)-1-methyl-pyrrolidin-2-ylmethoxy)-p...)
Affinity DataKi:  85nMAssay Description:Nicotinic acetylcholine receptor binding activity was determined by ability of the compound to displace [3H]- (-) cytisine binding from whole rat bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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