Reaction Details Report a problem with these data
Target
Protein mono-ADP-ribosyltransferase PARP16 [1-280]
Ligand
BDBM199181
Substrate
n/a
Meas. Tech.
Enzymatic Activity Assay
IC50
4.17e+3±n/a nM
Citation
Venkannagari, H; Verheugd, P; Koivunen, J; Haikarainen, T; Obaji, E; Ashok, Y; Narwal, M; Pihlajaniemi, T; Lüscher, B; Lehtiö, L Small-Molecule Chemical Probe Rescues Cells from Mono-ADP-Ribosyltransferase ARTD10/PARP10-Induced Apoptosis and Sensitizes Cancer Cells to DNA Damage. Cell Chem Biol 23:1251-1260 (2016) [PubMed] Article
More Info.:
Target
Name:
Protein mono-ADP-ribosyltransferase PARP16 [1-280]
Synonyms:
ARTD15 | C15orf30 | Human diphtheria toxin-like ADP-ribosyltransferase (ARTD15 or PARP16) | PAR16_HUMAN | PARP16
Type:
n/a
Mol. Mass.:
31385.07
Organism:
Homo sapiens (Human)
Description:
Q8N5Y8 (1-280 aa)
Residue:
280
Sequence:
MQPSGWAAAREAAGRDMLAADLRCSLFASALQSYKRDSVLRPFPASYARGDCKDFEALLADASKLPNLKELLQSSGDNHKRAWDLVSWILSSKVLTIHSAGKAEFEKIQKLTGAPHTPVPAPDFLFEIEYFDPANAKFYETKGERDLIYAFHGSRLENFHSIIHNGLHCHLNKTSLFGEGTYLTSDLSLALIYSPHGHGWQHSLLGPILSCVAVCEVIDHPDVKCQTKKKDSKEIDRRRARIKHSEGGDIPPKYFVVTNNQLLRVKYLLVYSQKPPKRAS