Reaction Details Report a problem with these data
Target
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q]
Ligand
BDBM214800
Substrate
n/a
Meas. Tech.
[35S]GTPγS Binding/Immunoprecipitation Assay
Kd
0.44±0.08 nM
Citation
Hu, J; Hu, K; Liu, T; Stern, MK; Mistry, R; Challiss, RA; Costanzi, S; Wess, J Novel structural and functional insights into M3 muscarinic receptor dimer/oligomer formation. J Biol Chem 288:34777-90 (2013) [PubMed] Article
More Info.:
Target
Name:
Muscarinic acetylcholine receptor M3 [1-273,470-589,N6Q,N15Q,N41Q,N48Q,N52Q]
Synonyms:
ACM3_RAT | Chrm-3 | Chrm3 | M3 muscarinic receptor (M3'(3C)-Xa)
Type:
Protein
Mol. Mass.:
46046.63
Organism:
Rattus norvegicus (Rat)
Description:
Modified rat M3R Δ274-469 lacking N-glycosylation sites (N6Q, N15Q, N41Q, N48Q, N52Q) and contains triple factor Xa site (IEGR)3 within i3 loop
Residue:
405
Sequence:
MTLHSQSTTSPLFPQISSSWVHSPSEAGLPLGTVTQLGSYQISQETGQFSSQDTSSDPLGGHTIWQVVFIAFLTGFLALVTIIGNILVIVAFKVNKQLKTVNNYFLLSLACADLIIGVISMNLFTTYIIMNRWALGNLACDLWLSIDYVASNASVMNLLVISFDRYFSITRPLTYRAKRTTKRAGVMIGLAWVISFVLWAPAILFWQYFVGKRTVPPGECFIQFLSEPTITFGTAIAAFYMPVTIMTILYWRIYKETEKRTKELAGLQASGTEIEGRIEGRIEGRTRSQITKRKRMSLIKEKKAAQTLSAILLAFIITWTPYNIMVLVNTFCDSCIPKTYWNLGYWLCYINSTVNPVCYALCNKTFRTTFKTLLLCQCDKRKRRKQQYQQRQSVIFHKRVPEQAL