Reaction Details Report a problem with these data
Target
Apoptosis regulator Bcl-2
Ligand
BDBM238186
Substrate
n/a
Meas. Tech.
Fluorescence Polarization-Based Binding Assay
pH
7.4±n/a
Temperature
298.15±n/a K
Ki
>4000±n/a nM
Comments
extracted
Citation
Nikolovska-Coleska, Z; Abulwerdi, F; Showalter, H; Miao, L; Stuckey, J; Mady, A Small molecule inhibitors of MCL-1 and uses thereof US Patent US9394303 Publication Date 7/19/2016
More Info.:
Target
Name:
Apoptosis regulator Bcl-2
Synonyms:
BCL2_MOUSE | Bcl-2 | Bcl2
Type:
Protein
Mol. Mass.:
26409.44
Organism:
Mus musculus (Mouse)
Description:
P10417
Residue:
236
Sequence:
MAQAGRTGYDNREIVMKYIHYKLSQRGYEWDAGDADAAPLGAAPTPGIFSFQPESNPMPAVHRDMAARTSPLRPLVATAGPALSPVPPVVHLTLRRAGDDFSRRYRRDFAEMSSQLHLTPFTARGRFATVVEELFRDGVNWGRIVAFFEFGGVMCVESVNREMSPLVDNIALWMTEYLNRHLHTWIQDNGGWDAFVELYGPSMRPLFDFSWLSLKTLLSLALVGACITLGAYLGHK