Reaction Details Report a problem with these data
Target
Resistance to inhibitors of cholinesterase protein 3
Ligand
BDBM82070
Substrate
n/a
Meas. Tech.
functional assay
EC50
6210±560 nM
Citation
Martin, RJ; Robertson, AP; VanVeller, B; Du, X; Zheng, F (S)-5-ethynyl-anabasine, derivatives thereof, and related compositions and methods of making and using US Patent US10667515 Publication Date 6/2/2020
More Info.:
Target
Name:
Resistance to inhibitors of cholinesterase protein 3
Synonyms:
F1L1D9_ASCSU
Type:
Protein
Mol. Mass.:
39160.01
Organism:
Pig roundworm
Description:
F1L1D9
Residue:
346
Sequence:
MPNSETATRSRRRRRRSSDDDDGPVSGWKMGLVVGVVVLCFGMLYPSLFHPMISSFFSKPPPPQQTIPNRPPIHPSMSSPRARPDIHPGMRMAAAQAEATATSSSKGMFAWMLPLYTVGVVVFLIYTLVKSKRKKQRRRHAYSSDESESYGEDDEYEQRGPGVHNLGRRKLRSLQERLKQTELAMSKILEQLGTISVDPTQGTVPQNLENTVDQKSKTNGESKKADVDKEHYLRDLEKALREFKHLSNSYNKEERKRRGESLSEEEEMNEDEFEEEMDEDEGTEEKSHGGGGSAGSAAEDEAENCSEDEREEKQEDDGKKGEDEVLVPAVEQHVQQTKPHKRSKRT