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TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353018(CHEMBL1821980 | CHEMBL1852660)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of human APNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025070(CHEMBL3355110)
Affinity DataKi:  0.210nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353018(CHEMBL1821980 | CHEMBL1852660)
Affinity DataKi:  0.350nMAssay Description:Inhibition of human APN using L-leucine-p-nitroanilide as substrate measured every 10 mins for 2 hrs by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025066(CHEMBL3355109)
Affinity DataKi:  0.690nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 1nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025099(CHEMBL3355111)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025041(CHEMBL3355106)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025043(CHEMBL3355104)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  2nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025042(CHEMBL3355105)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025050(CHEMBL3355108)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50393210(CHEMBL1235787)
Affinity DataKi:  2.20nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025046(CHEMBL3355101)
Affinity DataKi:  2.40nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105262(2-{3-[(1-Amino-ethyl)-hydroxy-phosphinoyl]-2-biphe...)
Affinity DataKi:  2.90nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, aminopeptidase N(APN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50528308(CHEMBL4460082)
Affinity DataKi:  4.5nMAssay Description:Inhibition of soluble human APN ectodomain stably expressed in HEK293 GnTI(-) cells using H-Leu-NHMec as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50025047(CHEMBL3355100)
Affinity DataKi:  4.80nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105263(2-{3-[(Amino-phenyl-methyl)-hydroxy-phosphinoyl]-2...)
Affinity DataKi:  4.80nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, aminopeptidase N(APN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of human recombinant alanyl aminopeptidase after 30 to 60 mins by morrison's equationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataKi:  8nMAssay Description:Inhibition of APN in human placenta using AlabetaNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50078133(2-Amino-4-methyl-pentane-1-thiol | (S)-2-Amino-4-m...)
Affinity DataIC50: 8nMAssay Description:Inhibition of FLAG-tagged human recombinant Aminopeptidase NMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50528311(CHEMBL4448936)
Affinity DataKi:  8.20nMAssay Description:Inhibition of soluble human APN ectodomain stably expressed in HEK293 GnTI(-) cells using H-Leu-NHMec as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50415629(CHEMBL1077583)
Affinity DataKi:  8.51nMAssay Description:Inhibition of catalytic activity of human aminopeptidase N transfected in HEK293 cells assessed as formation of p-nitroanilineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50023134(CHEMBL3298943)
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human Aminopeptidase N using L-Ala-beta-NA as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50023133(CHEMBL3298942)
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant human Aminopeptidase N using L-Ala-beta-NA as substrate preincubated for 30 mins followed by substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2016
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50023133(CHEMBL3298942)
Affinity DataKi:  11nMAssay Description:Inhibition of human recombinant APN using L-Ala-beta-NA as substrate after 30 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50353016(CHEMBL1821978)
Affinity DataKi:  11nMAssay Description:Inhibition of human APN using L-leucine-p-nitroanilide as substrate measured every 10 mins for 2 hrs by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50023134(CHEMBL3298943)
Affinity DataKi:  11nMAssay Description:Inhibition of human recombinant APN using L-Ala-beta-NA as substrate after 30 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataIC50: 11nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50105261(benzyl 2-[(2S)-2-({[(2S)-2-azaniumyl-4-(methylsulf...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for inhibition of enkephalin degrading enzyme, aminopeptidase N(APN)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50415628(CHEMBL1077582)
Affinity DataKi:  12.6nMAssay Description:Inhibition of catalytic activity of human aminopeptidase N transfected in HEK293 cells assessed as formation of p-nitroanilineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50023135(CHEMBL3298944)
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant APN using L-Ala-beta-NA as substrate after 30 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50528345(CHEMBL4445188)
Affinity DataKi:  19nMAssay Description:Inhibition of soluble human APN ectodomain stably expressed in HEK293 GnTI(-) cells using H-Leu-NHMec as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457485(CHEMBL4205440)
Affinity DataKi:  19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457467(CHEMBL4217873)
Affinity DataKi:  19nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50435737(PROBESTIN)
Affinity DataKi:  19nMAssay Description:Inhibition of aminopeptidase N (unknown origin) using L-leucine-beta-naphthylamide as substrate after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457478(CHEMBL4208547)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457468(CHEMBL4216928)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50368599(CHEMBL1159809)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457477(CHEMBL4210855)
Affinity DataKi:  20nMAssay Description:Inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50457471(CHEMBL1159811)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50368598(CHEMBL1159810)
Affinity DataIC50: 21nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase N(Human)
University of Upper Alsace

Curated by ChEMBL
LigandPNGBDBM50528319(CHEMBL4566015)
Affinity DataKi:  23nMAssay Description:Inhibition of soluble human APN ectodomain stably expressed in HEK293 GnTI(-) cells using H-Leu-NHMec as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
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