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Report error Found 12 of affinity data for UniProtKB/TrEMBL: P16615
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50527071(CHEMBL4514624)
Affinity DataKi:  1.30nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50453611(CHEMBL4207081)
Affinity DataKi:  11nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50631114(CHEMBL5435124)
Affinity DataEC50:  16nMAssay Description:Activation of SERCA2a in human HEK293T cells endoplasmic reticulum assessed as increase in calcium release measured for 10 mins in presence of ATP by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  23nMAssay Description:Binding affinity to human ATP2A2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50453612(CHEMBL4216774)
Affinity DataKi:  27nMAssay Description:Inhibition of SERCA2a (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50527068(CHEMBL468766 | CHEBI:17734)
Affinity DataIC50: 90nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50527063(CHEMBL4534285)
Affinity DataIC50: 210nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM176764(US9688816, 7 | 2,5-Di-tert-butylhydroquinone | CAS...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50854(MLS000028812 | SMR000058863 | PAXILLINE | cid_1050...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of SERCA2b in human platelet microsomes by enzyme-coupled methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  9.67E+3nMAssay Description:Binding affinity to human ATP2A2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Human)
University of Chemistry and Technology Prague

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition of human SERCA2b expressed in COS7 cells microsomal membranes preincubated for 10 mins followed by addition of ATP and measured after 40 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed