Compile Data Set for Download or QSAR
Report error Found 581 of affinity data for UniProtKB/TrEMBL: P31389
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50017721(5-(1-methylpiperidylidene-4)-5H-dibenzo(a,d)cyclop...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002099(CHEMBL366965 | Dimethyl-[3-(2-methyl-6H-dibenzo[b,...)
Affinity DataKi:  0.130nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50079527(CHEMBL101740 | cis-doxepin | DOXEPIN | (3E)-3-dibe...)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50020712(CHEMBL629 | Amitriptylin | 10,11-dihydro-N,N-dimet...)
Affinity DataKi:  0.170nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50007538(CHEMBL25626 | 8-(2-Azetidin-1-yl-ethyl)-3-chloro-6...)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of [3H]mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50079527(CHEMBL101740 | cis-doxepin | DOXEPIN | (3E)-3-dibe...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50292411(Actahist | CHEMBL855 | Actifed | Myfed | Triphed |...)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002087(4-(1-Methyl-piperidin-4-ylidene)-4,9-dihydro-1-thi...)
Affinity DataKi:  0.310nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  0.440nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002083(CHEMBL65612 | 2-[11-(3-Dimethylamino-propylidene)-...)
Affinity DataKi:  0.480nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  0.570nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86032(trans-PAT | trans-H2-PAT(-))
Affinity DataKi:  0.580nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002102(CHEMBL294777 | 2-[11-(3-Dimethylamino-propylidene)...)
Affinity DataKi:  0.630nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50292411(Actahist | CHEMBL855 | Actifed | Myfed | Triphed |...)
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM24226(cid_2247 | [3H]-ASTEMIZOLE | Hismanal | ASTEMIZOLE...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKd:  0.851nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM84994(NSC_163091 | CAS_163091 | ORG-5222)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50292411(Actahist | CHEMBL855 | Actifed | Myfed | Triphed |...)
Affinity DataKi:  0.930nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86174(CAS_486-12-4 | NSC_5282443 | Triprolidine)
Affinity DataKi:  0.930nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86032(trans-PAT | trans-H2-PAT(-))
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86174(CAS_486-12-4 | NSC_5282443 | Triprolidine)
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86032(trans-PAT | trans-H2-PAT(-))
Affinity DataKi:  1.15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  1.23nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  1.37nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22567(CHEMBL511 | PYRILAMINE | 3H]pyrilamine | N-[2-(dim...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of guinea pig histamine H1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86033(cis-H2-PAT(+/-) | trans-H2-PAT(+/-))
Affinity DataKi:  1.53nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50131441(9,13b-dihydro-1H-dibenzo[c,f]imidazo[1,5-a]azepin-...)
Affinity DataIC50: 1.58nMAssay Description:Potency against histamine H1 receptor on guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50007542(CHEMBL24835 | 3-Chloro-8-(2-dimethylamino-ethyl)-6...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of [3H]mepyramine binding to the histamine receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM35938(clorfeniramina | gamma-(4-chlorophenyl)-N,N-dimeth...)
Affinity DataKi:  1.98nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  2.07nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM35255(2-Chloro-11-(2-(dimethylamino)ethoxy)dibenzo(b,f)t...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50509922(CHEMBL4575319)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-mepyramine from histamine H1 receptor in guinea pig cerebellum homogenates incubated for 60 mins by Cheng and Prusoff equation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50419322(CHEMBL1910386)
Affinity DataKd:  3.80nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]mepyramine from histamine H1 receptor in guinea pig cerebellum after 60 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM24226(cid_2247 | [3H]-ASTEMIZOLE | Hismanal | ASTEMIZOLE...)
Affinity DataKd:  3.80nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86031(cis-H2-PAT(-))
Affinity DataKi:  3.92nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002103(CHEMBL293652 | 3-[11-(3-Dimethylamino-propylidene)...)
Affinity DataKi:  4.20nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002095(CHEMBL65822 | 11-(3-Dimethylamino-propylidene)-6,1...)
Affinity DataKi:  4.20nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002085(CHEMBL304185 | [11-(4-Dimethylamino-butylidene)-6,...)
Affinity DataKi:  4.60nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50419326(CHEMBL1910381)
Affinity DataKd:  4.90nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM86031(cis-H2-PAT(-))
Affinity DataKi:  4.91nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002086(CHEMBL304223 | 11-(3-Pyrrolidin-1-yl-propylidene)-...)
Affinity DataKi:  5nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetHistamine H1 receptor(Guinea pig)
UniversitÉ

Curated by PDSP Ki Database
LigandPNGBDBM50002093(CHEMBL65699 | [11-(3-Dimethylamino-propylidene)-6,...)
Affinity DataKi:  5.20nMAssay Description:The compound was tested in vitro for binding affinity against histamine H1 receptor from guinea pig cerebellum, using [3H]pyrilamine as radioligand a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 581 total ) | Next | Last >>
Jump to: