Compile Data Set for Download or QSAR
Report error Found 680 of affinity data for UniProtKB/TrEMBL: P56450
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50158406(Ac-Nle-c[Asp-His-DPhe-Arg-Trp-Lys]-NH2 | CHEMBL224...)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031473(CHEMBL3358549)
Affinity DataEC50:  0.0480nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at mouse melanocortin-4 receptor transfected in HEK293 cells after 6 hrs by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/29/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031479(CHEMBL3358545)
Affinity DataEC50:  0.0510nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50410399(CHEMBL2096712)
Affinity DataEC50:  0.0530nMAssay Description:Effective concentration for mouse Melanocortin-4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031488(CHEMBL3358541)
Affinity DataEC50:  0.0580nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  0.0600nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50166123([(2S,5R,8R,11R,14S,17R)-1-(2-Acetylamino-hexanoyl)...)
Affinity DataEC50:  0.0600nMAssay Description:In vitro agonist potency for Mouse Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031469(CHEMBL3358552)
Affinity DataEC50:  0.0670nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  0.0870nMAssay Description:Activity in mouse melanocortin-4 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50114736([1-(2-Acetylamino-hexanoyl)-17-(4-amino-butyl)-8-b...)
Affinity DataEC50:  0.0870nMAssay Description:In vitro activation of mouse recombinant Melanocortin-4 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50184359(MT-II | CHEMBL430239 | Ac-Nle-c[Asp-His-DPhe-Arg-T...)
Affinity DataEC50:  0.0870nMAssay Description:Agonist activity to the mouse Melanocortin-4 receptor (mMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50144873(Ac-Nle-c[Asp-His-DPhe-Arg-Trp-Gly-Lys]-NH2 | CHEMB...)
Affinity DataEC50:  0.0870nMAssay Description:Effective concentration against mouse melanocortin MC4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.0970nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031492(CHEMBL3358539)
Affinity DataEC50:  0.0980nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as stimulation of intracellular cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at mouse melanocortin-4 receptor expressed in HEK293 cells co-transfected with CRE/beta-galactosidase reporter gene assessed as stim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50410408(CHEMBL2096713)
Affinity DataEC50:  0.130nMAssay Description:Effective concentration for mouse Melanocortin-4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031496(CHEMBL3358535)
Affinity DataEC50:  0.130nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.140nMAssay Description:In vitro agonist potency for Mouse Melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031478(CHEMBL3358546)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031471(CHEMBL3358550)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50499283(CHEMBL3735690)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at mouse MC4 receptor expressed in HEK293 cells after 2 hrs by cAMP alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.140nMAssay Description:Agonistic activity against mouse MC4RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031470(CHEMBL3358551)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031490(CHEMBL3358540)
Affinity DataEC50:  0.140nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50499283(CHEMBL3735690)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at mouse MC4 receptor expressed in HEK293 cells after 2 hrs by cAMP alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.160nMAssay Description:Effective concentration for mouse Melanocortin-4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50339348((4R,7S,10S,13S,16S,19S,22R,25S,28R)-25-((1H-imidaz...)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at mouse MC4 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50144869(Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-Phe-Dpr]-Tyr-NH...)
Affinity DataEC50:  0.180nMAssay Description:Effective concentration against mouse melanocortin MC4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031495(CHEMBL3358536)
Affinity DataEC50:  0.190nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at mouse MC4 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.200nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50141023(1N-(1-carbamoyl-2-hydroxypropyl)-15-[3-amino(imino...)
Affinity DataEC50:  0.200nMAssay Description:Effective concentration for maximum agonist response towards mouse melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.210nMAssay Description:Effective concentration against mouse melanocortin MC4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.210nMAssay Description:In vitro activation of mouse recombinant Melanocortin-4 receptor.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity to the mouse Melanocortin-4 receptor (mMC4R)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031500(CHEMBL2372859)
Affinity DataEC50:  0.210nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataEC50:  0.210nMAssay Description:Activity in mouse melanocortin-4 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031486(CHEMBL3358544)
Affinity DataEC50:  0.220nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50144869(Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-Phe-Dpr]-Tyr-NH...)
Affinity DataIC50: 0.260nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50410403(CHEMBL2096717)
Affinity DataEC50:  0.270nMAssay Description:Effective concentration for mouse Melanocortin-4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50339348((4R,7S,10S,13S,16S,19S,22R,25S,28R)-25-((1H-imidaz...)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.279nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells co-expressing CRE/beta-galactosidase reporter gene after 6 hrs by beta-galactosidase cAMP as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.290nMAssay Description:Effective concentration for maximum agonist response towards mouse melanocortin 4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50031489(CHEMBL3352878)
Affinity DataEC50:  0.290nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
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