Compile Data Set for Download or QSAR
Report error Found 203 for UniProtKB: Q9HBW0
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50056344BDBM50056344(CHEMBL3322514)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50056343BDBM50056343(CHEMBL3322513)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50594511BDBM50594511(CHEMBL5182278)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to LPA2 receptor (unknown origin) by free solution assay-compensated interferometric reader (FSA-CIR) techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50557594BDBM50557594(CHEMBL4788435 | US11485727, Example 1.3 | US202600...)
Affinity DataIC50: 1.5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50557595BDBM50557595(CHEMBL4745566 | US11485727, Example 1.7 | US202600...)
Affinity DataIC50: 1.60nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50557597BDBM50557597(CHEMBL4758133 | US11485727, Example 2.6 | US202600...)
Affinity DataIC50: 1.80nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50557599BDBM50557599(CHEMBL4751395 | US11485727, Example 2.10 | US20260...)
Affinity DataIC50: 1.80nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50557598BDBM50557598(CHEMBL4784419 | US11485727, Example 2.7 | US202600...)
Affinity DataIC50: 1.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50557596BDBM50557596(CHEMBL4743845 | US11485727, Example 2.4 | US202600...)
Affinity DataIC50: 1.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50148348BDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579837BDBM579837(US11485727, Example 2.8 | US20260001863, Example 2...)
Affinity DataIC50: 2nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 191570BDBM191570(US9670204, 12 2-((2-ethyl-8-fluoro-6-(4-(2-(3-hydr...)
Affinity DataIC50: 2nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 50285777BDBM50285777(CHEMBL4165749 | BI-2545 (19) | ACS Med. Chem. Lett...)
Affinity DataIC50: 2.20nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579844BDBM579844(US11485727, Example 2.15 | US20260001863, Example ...)
Affinity DataIC50: 2.20nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579832BDBM579832(US11485727, Example 2.3 | US20260001863, Example 2...)
Affinity DataIC50: 2.20nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 97150BDBM97150(N-methyl-N-[1-(4-{[(6-{[6-(trifluoromethyl)pyridin...)
Affinity DataIC50: 2.30nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579848BDBM579848(US11485727, Example 2.19 | US20260001863, Example ...)
Affinity DataIC50: 2.40nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579850BDBM579850(US11485727, Example 2.21 | US20260001863, Example ...)
Affinity DataIC50: 2.40nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579834BDBM579834(US11485727, Example 2.5 | US20260001863, Example 2...)
Affinity DataIC50: 2.5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579853BDBM579853(1-[4-(4-{[(6-{[6-(Difluoromethyl)pyridin-3-yl]meth...)
Affinity DataIC50: 2.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579824BDBM579824(US11485727, Example 1.2 | US20260001863, Example 1...)
Affinity DataIC50: 2.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579849BDBM579849(US11485727, Example 2.20 | US20260001863, Example ...)
Affinity DataIC50: 2.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50233165BDBM50233165(CHEMBL1222042)
Affinity DataEC50:  3nMAssay Description:Agonist activity at LPA2 receptor (unknown origin) expressed in MEF cells assessed as increase in intracellular calcium level measured every 3.42 sec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2019
Entry Details Article
PubMed
TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579831BDBM579831(US11485727, Example 2.2 | US20260001863, Example 2...)
Affinity DataIC50: 3nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579826BDBM579826(US11485727, Example 1.4 | US20260001863, Example 1...)
Affinity DataIC50: 3.30nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579823BDBM579823(3-{[6-(Difluoromethyl)pyridin-3-yl]methoxy}-6-iodo...)
Affinity DataIC50: 3.40nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579841BDBM579841(US11485727, Example 2.12 | US20260001863, Example ...)
Affinity DataIC50: 3.5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579838BDBM579838(US11485727, Example 2.9 | US20260001863, Example 2...)
Affinity DataIC50: 3.70nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579840BDBM579840(US11485727, Example 2.11 | US20260001863, Example ...)
Affinity DataIC50: 3.80nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579852BDBM579852(US11485727, Example 2.23 | US20260001863, Example ...)
Affinity DataIC50: 3.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579827BDBM579827(US11485727, Example 1.5 | US20260001863, Example 1...)
Affinity DataIC50: 3.90nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579842BDBM579842(US11485727, Example 2.13 | US20260001863, Example ...)
Affinity DataIC50: 4nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579843BDBM579843(US11485727, Example 2.14 | US20260001863, Example ...)
Affinity DataIC50: 4.40nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 719985BDBM719985(US20250051321, Compound GLPG1690 | WO2014139882, C...)
Affinity DataIC50: 5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579846BDBM579846(US11485727, Example 2.17 | US20260001863, Example ...)
Affinity DataIC50: 5.20nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579851BDBM579851(US11485727, Example 2.22 | US20260001863, Example ...)
Affinity DataIC50: 6.20nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579828BDBM579828(US11485727, Example 1.6 | US20260001863, Example 1...)
Affinity DataIC50: 6.5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50148435BDBM50148435([3-(3,5-Dichloro-4-octyloxy-benzylamino)-propyl]-p...)
Affinity DataIC50: 6.60nMAssay Description:Binding affinity to human sphingosine 1-phosphate receptor 4 expressed in CHO cells was determined by using [33P]-S1P as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50148348BDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  6.80nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579855BDBM579855(1-((3aR,3bS,6aR,6bS)-5-(4-(((6-((6-(trifluoromethy...)
Affinity DataIC50: 7nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50271765BDBM50271765(4,4'-(4,4'-(1,3-phenylenebis(oxy))bis(4,1-phenylen...)
Affinity DataKi:  7.20nMAssay Description:Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579854BDBM579854(1-[(3aR,8aS)-2-(4-{[(6-{[6-(trifluoromethyl)pyridi...)
Affinity DataIC50: 8.60nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50271765BDBM50271765(4,4'-(4,4'-(1,3-phenylenebis(oxy))bis(4,1-phenylen...)
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50271765BDBM50271765(4,4'-(4,4'-(1,3-phenylenebis(oxy))bis(4,1-phenylen...)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAutotaxin/Lysophosphatidic acid receptor 2(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 579847BDBM579847(US11485727, Example 2.18 | US20260001863, Example ...)
Affinity DataIC50: 9.20nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Confirmation testing of small molecules identifie...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2026
Entry Details
US Patent

TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610664BDBM50610664(CHEMBL5283300)
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610665BDBM50610665(CHEMBL5290275)
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610663BDBM50610663(CHEMBL5282947)
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610666BDBM50610666(CHEMBL5278054)
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50610667BDBM50610667(CHEMBL5266099)
Affinity DataIC50: 10nMAssay Description:Inhibition of LPA2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
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