Compile Data Set for Download or QSAR
Report error Found 543 for UniProtKB: Q9NS75
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227045BDBM50227045(CHEMBL354129)
Affinity DataIC50: 0.0310nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50023198BDBM50023198(CHEMBL21333 | N-(4-oxo-2-(1H-tetrazol-5-yl)-4H-chr...)
Affinity DataIC50: 0.0440nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227075BDBM50227075(CHEMBL171021)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227363BDBM50227363(CHEMBL299837)
Affinity DataKi:  0.100nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227072BDBM50227072(CHEMBL169790)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227054BDBM50227054(CHEMBL354530)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227053BDBM50227053(CHEMBL170191)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069352BDBM50069352((1-{(R)-1-{3-[(E)-2-(7,7-Dimethyl-5,6,7,8-tetrahyd...)
Affinity DataIC50: 0.170nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069356BDBM50069356([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 0.190nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069352BDBM50069352((1-{(R)-1-{3-[(E)-2-(7,7-Dimethyl-5,6,7,8-tetrahyd...)
Affinity DataIC50: 0.190nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50068974BDBM50068974(CGP-57698 | 2,2-Diethyl-N-[3-(7-fluoro-quinolin-2-...)
Affinity DataIC50: 0.200nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009075BDBM50009075(CHEMBL22033 | ICI 198615 | [1-(4-Benzenesulfonylam...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against cysteinyl leukotriene D4 receptor from guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227366BDBM50227366(CHEMBL48927)
Affinity DataKi:  0.200nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069375BDBM50069375((R)-2-(1-((1-(3-(2-(5,7-dihydrothieno[3,4-b]pyridi...)
Affinity DataIC50: 0.210nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227364BDBM50227364(CHEMBL299093)
Affinity DataKi:  0.25nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227361BDBM50227361(CHEMBL51585)
Affinity DataKi:  0.25nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215369BDBM50215369(CHEMBL368290)
Affinity DataIC50: 0.300nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227642BDBM50227642(CHEMBL50562)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227358BDBM50227358(CHEMBL412056)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227356BDBM50227356(CHEMBL49944)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227365BDBM50227365(CHEMBL300096)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227355BDBM50227355(CHEMBL296821)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227640BDBM50227640(CHEMBL297952)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50066948BDBM50066948(CHEMBL3403187)
Affinity DataIC50: 0.310nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069372BDBM50069372((1-{(R)-1-{3-[(E)-2-(6,6-Dimethyl-6,7-dihydro-5H-[...)
Affinity DataIC50: 0.340nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069350BDBM50069350((1-{(R)-1-{3-[(E)-2-(7,7-Dimethyl-6,7-dihydro-5H-[...)
Affinity DataIC50: 0.350nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227047BDBM50227047(CHEMBL172889)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215411BDBM50215411(CHEMBL425675)
Affinity DataIC50: 0.400nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069372BDBM50069372((1-{(R)-1-{3-[(E)-2-(6,6-Dimethyl-6,7-dihydro-5H-[...)
Affinity DataIC50: 0.430nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052024BDBM50052024(montelukast | CHEMBL787)
Affinity DataIC50: 0.430nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227136BDBM50227136(CHEMBL170100)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50066911BDBM50066911(CHEMBL3401689)
Affinity DataIC50: 0.490nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069355BDBM50069355((R)-2-(1-((1-(3-(2-(6,7-dihydro-5H-cyclopenta[b]py...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227390BDBM50227390(CHEMBL301616)
Affinity DataKi:  0.5nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215410BDBM50215410(CHEMBL369421)
Affinity DataIC50: 0.5nMAssay Description:In vitro for antagonistic activity against LTD4 receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069364BDBM50069364((R)-2-(1-((1-(3-(2-(6-butyl-5-methylpyridin-2-yl)v...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227144BDBM50227144(CHEMBL83797)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216211BDBM50216211(CHEMBL143597)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069373BDBM50069373(2-(1-(((1R)-3-(2-(2-hydroxypropan-2-yl)phenyl)-1-(...)
Affinity DataIC50: 0.510nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069357BDBM50069357([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 0.580nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033089BDBM50033089(CHEMBL3342959)
Affinity DataIC50: 0.620nMAssay Description:Antagonist activity at human CysLT2 receptor expressed in HEK293 cells assessed as inhibition of LTD4-inudced intracellular calcium influx preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2016
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069373BDBM50069373(2-(1-(((1R)-3-(2-(2-hydroxypropan-2-yl)phenyl)-1-(...)
Affinity DataIC50: 0.630nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052024BDBM50052024(montelukast | CHEMBL787)
Affinity DataIC50: 0.640nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227063BDBM50227063(CHEMBL170017)
Affinity DataIC50: 0.670nMAssay Description:Inhibition of LTC4 induced smooth muscle contraction of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216211BDBM50216211(CHEMBL143597)
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50227389BDBM50227389(CHEMBL51580)
Affinity DataKi:  0.700nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069354BDBM50069354([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 0.730nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069370BDBM50069370((1-{(R)-1-{3-[(E)-2-(2,3-Dihydro-thieno[3,2-b]pyri...)
Affinity DataIC50: 0.740nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069371BDBM50069371((1-{(R)-1-{3-[(E)-2-(8,8-Dimethyl-5,6,7,8-tetrahyd...)
Affinity DataIC50: 0.75nMAssay Description:In vitro inhibition of [3H]LTD4 binding to LTD4 receptor of guinea pig lung membrane with human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1/2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50216210BDBM50216210(CHEMBL141234)
Affinity DataIC50: 0.800nMAssay Description:In vitro inhibition of [3H]-LTD4 binding to LTD4 receptor of guinea pig lung membrane without human serum albumin (HSA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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