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Phenolic compounds with pancreatic lipase inhibitory activity from Korean yam (Dioscorea opposita).BDB
J Enzyme Inhib Med Chem 29: 1-6 (2014)
Seoul National University
Synthesis and carbonic anhydrase inhibitory properties of novel 1,4-dihydropyrimidinone substituted diarylureas.BDB
J Enzyme Inhib Med Chem 29: 18-22 (2014)
Sakarya University
Carbonic anhydrase inhibitory properties of novel sulfonamide derivatives of aminoindanes and aminotetralins.BDB
J Enzyme Inhib Med Chem 29: 35-42 (2014)
Atatürk University
Phenolic phytochemical displaying SARS-CoV papain-like protease inhibition from the seeds of Psoralea corylifolia.BDB
J Enzyme Inhib Med Chem 29: 59-63 (2014)
Gyeongsang National University
In vitro inhibition effect and structure-activity relationships of some saccharin derivatives on erythrocyte carbonic anhydrase I and II.BDB
J Enzyme Inhib Med Chem 29: 118-23 (2014)
Sakarya University
Benzenesulfonamides with benzimidazole moieties as inhibitors of carbonic anhydrases I, II, VII, XII and XIII.BDB
J Enzyme Inhib Med Chem 29: 124-31 (2014)
Vilnius University
Synthesis and carbonic anhydrase inhibitory properties of 1,3-dicarbonyl derivatives of methylaminobenzene-sulfonamide.BDB
J Enzyme Inhib Med Chem 29: 132-6 (2014)
Sakarya University
Synthesis and carbonic anhydrase isoenzymes I and II inhibitory effects of novel benzylamine derivatives.BDB
J Enzyme Inhib Med Chem 29: 168-74 (2014)
Atatürk University
Antileishmanial activity evaluation of bis-lawsone analogs and DNA topoisomerase-I inhibition studies.BDB
J Enzyme Inhib Med Chem 29: 185-9 (2014)
Karunya University
New chemotypes as Trypanosoma cruzi triosephosphate isomerase inhibitors: a deeper insight into the mechanism of inhibition.BDB
J Enzyme Inhib Med Chem 29: 198-204 (2014)
Universidad De La Republica
Discovery of new HER2/EGFR dual kinase inhibitors based on the anilinoquinazoline scaffold as potential anti-cancer agents.BDB
J Enzyme Inhib Med Chem 29: 215-22 (2014)
Msa University
Cytotoxicity and topoisomerase I/II inhibition activity of novel 4-aryl/alkyl-1-(piperidin-4-yl)-carbonylthiosemicarbazides and 4-benzoylthiosemicarbazides.BDB
J Enzyme Inhib Med Chem 29: 243-8 (2014)
Medical University
Synthesis and evaluation of 18F-labeled carbonic anhydrase IX inhibitors for imaging with positron emission tomography.BDB
J Enzyme Inhib Med Chem 29: 249-55 (2014)
Bc Cancer Agency
Synthesis and dual D2 and 5-HT1A receptor binding affinities of 5-piperidinyl and 5-piperazinyl-1H-benzo[d]imidazol-2(3H)-ones.BDB
J Enzyme Inhib Med Chem 29: 281-91 (2014)
King Fahd University of Petroleum & Minerals
Novel coumarins and benzocoumarins acting as isoform-selective inhibitors against the tumor-associated carbonic anhydrase IX.BDB
J Enzyme Inhib Med Chem 29: 292-6 (2014)
S.G.S.I.T.S.
Novel inhibitor of bacterial sphingomyelinase, SMY-540, developed based on three-dimensional structure analysis.BDB
J Enzyme Inhib Med Chem 29: 303-10 (2014)
Tokushima Bunri University
Design, synthesis and evaluation of 2-phenylisothiazolidin-3-one-1,1-dioxides as a new class of human protein kinase CK2 inhibitors.BDB
J Enzyme Inhib Med Chem 29: 338-43 (2014)
Nas of Ukraine
Design, synthesis and biological evaluation of novel inosine 5'-monophosphate dehydrogenase (IMPDH) inhibitors.BDB
J Enzyme Inhib Med Chem 29: 408-19 (2014)
Nycomed
Inhibition of mammalian carbonic anhydrases I-XIV with grayanotoxin III: solution and in silico studies.BDB
J Enzyme Inhib Med Chem 29: 469-75 (2014)
University of Calgary
Carbonic anhydrase inhibitors. Phenols incorporating 2- or 3-pyridyl-ethenylcarbonyl and tertiary amine moieties strongly inhibit Saccharomyces cerevisiae ß-carbonic anhydrase.BDB
J Enzyme Inhib Med Chem 29: 495-9 (2014)
Ataturk University
Biochemical characterization of the chloroplastic ß-carbonic anhydrase from Flaveria bidentis (L.) "Kuntze".BDB
J Enzyme Inhib Med Chem 29: 500-4 (2014)
Istituto Di Biostrutture E Bioimmagini-Cnr
Effects of novel human cathepsin S inhibitors on cell migration in human cancer cells.BDB
J Enzyme Inhib Med Chem 29: 538-46 (2014)
National Tsing Hua University
Identification and structure-activity relationship study of carvacrol derivatives as Mycobacterium tuberculosis chorismate mutase inhibitors.BDB
J Enzyme Inhib Med Chem 29: 547-54 (2014)
Birla Institute of Technology
Quinolone-based HDAC inhibitors.BDB
J Enzyme Inhib Med Chem 29: 555-62 (2014)
Orchid Chemicals & Pharmaceuticals
A systematic quantitative approach to rational drug design and discovery of novel human carbonic anhydrase IX inhibitors.BDB
J Enzyme Inhib Med Chem 29: 571-81 (2014)
Birla Institute of Technology
Discovery of a series of hydroximic acid derivatives as potent histone deacetylase inhibitors.BDB
J Enzyme Inhib Med Chem 29: 582-9 (2014)
Qingdao University