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Found 216 with Last Name = 'al-horani' and Initial = 'ra'
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608714(CHEMBL5281897)
Affinity DataIC50:  26nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608719(CHEMBL5269766)
Affinity DataIC50:  29nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human plasma coagulation factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608720(CHEMBL5285085)
Affinity DataIC50:  102nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM577548(US11472838, Compound Ref. 22)
Affinity DataIC50:  110nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608718(CHEMBL5286758)
Affinity DataIC50:  139nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50136842(CHEMBL152117 | GNF-Pf-5230 | N-[2-(4-Hydroxy-pheny...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human coagulation factor XIIIaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386271(CHEMBL2040983)
Affinity DataIC50:  270nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608713(CHEMBL5275210)
Affinity DataIC50:  310nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608710(CHEMBL5290263)
Affinity DataIC50:  350nMAssay Description:Inhibition of human plasma coagulation factor XIIIaMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50425968(CHEMBL2314388)
Affinity DataIC50:  551nMAssay Description:Inhibition of human FXIa assessed as S-2366 hydrolysis after 10 mins by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608712(CHEMBL5286863)
Affinity DataIC50:  610nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386267(CHEMBL2040979)
Affinity DataIC50:  900nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386261(CHEMBL2040973)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in absence of exosite 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386253(CHEMBL2040963)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455303(CHEMBL4218956)
Affinity DataIC50:  1.30E+3nMAssay Description:Partial allosteric inhibition of human thrombin using S-23666 as substrate measured after 1 min by fibrometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in absence of exosite 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386259(CHEMBL2040970)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 30 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386270(CHEMBL2040982)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 15 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  1.80E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain [Q652E](Homo sapiens (Human))TBA
LigandPNGBDBM50608711(CHEMBL5290280)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in absence of exosite 2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455292(CHEMBL4215598)
Affinity DataIC50:  2.00E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in absence of exosite 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455293(CHEMBL4208688)
Affinity DataIC50:  2.30E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455294(CHEMBL4203810)
Affinity DataIC50:  2.60E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455291(CHEMBL4214824)
Affinity DataIC50:  2.60E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455285(CHEMBL4207062)
Affinity DataIC50:  2.60E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 50 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 5 uM exo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 5 uM exo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 10 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50260048(CHEMBL4084933)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding affinity to human plasmin assessed as loss of intrinsic tryptophan fluorescence at 250 uM by spectrofluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 20 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 30 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50386266(CHEMBL2040978)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human factor 10a using chromogenic spectrozyme F10a as substrate after 10 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50608715(CHEMBL5273935)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of tissue transglutaminase (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455297(CHEMBL4218791)
Affinity DataIC50:  3.20E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455308(CHEMBL4203401)
Affinity DataIC50:  3.30E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 10 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455284(CHEMBL4210645)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 20 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  3.60E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50260048(CHEMBL4084933)
Affinity DataIC50:  3.60E+3nMAssay Description:Allosteric inhibition of human plasmin using chromogenic substrate spectrozyme PL preincubated for 5 mins followed by substrate addition measured ove...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455289(CHEMBL4212514)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition measured in presence of 15 uM ex...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455295(CHEMBL4214371)
Affinity DataIC50:  3.80E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50455307(CHEMBL4215073)
Affinity DataIC50:  4.00E+3nMAssay Description:Partial allosteric inhibition of human thrombin using spectrozyme TH as substrate pretreated for 10 mins followed by substrate addition by spectropho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50260048(CHEMBL4084933)
Affinity DataIC50:  4.60E+3nMAssay Description:Allosteric inhibition of human plasmin assessed as delay in clot lysis after 410 mins by spectrophotometer methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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