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Found 2334 with Last Name = 'sippl' and Initial = 'w'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50098203(1-{4-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-phenyl}-...)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [125I]-iodoproxyfan from rat histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132057(CHEMBL1180430 | CHEMBL126128 | N-{4-[4-(2-Methoxy-...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132040(3-(4-Methoxy-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pi...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50077001(1-Benzyl-4-(3-methyl-4-phenyl-pyrazol-1-yl)-piperi...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity of compound towards human Dopamine receptor D4 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132031(3-(4-Bromo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pipe...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132047(3-(4-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.440nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132060(3-(3-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132059(3-(4-Cyano-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pipe...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of human full length PKMYT1 expressed in HEK293 cells using EFS (247 to 259 residues) as substrate after 1 hr by fluorescence polarization...More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132012((E)-3-(4-Iodo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-p...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50506980(CHEMBL4583196)
Affinity DataKi:  0.5nMAssay Description:Displacement of (6-FAM)KI(pY)VV from full length PKMYT1 (unknown origin) by fluorescence polarization immuno assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132013(CHEMBL341542 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50007182(4-Chloro-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132027(3-(2-Chloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132076(3-Benzo[1,3]dioxol-4-yl-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  0.550nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132019(3-(2-Methoxy-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pi...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132070(CHEMBL338552 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132055(3-Furan-2-yl-N-{4-[4-(2-methoxy-phenyl)-piperazin-...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132039(CHEMBL126280 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132050(CHEMBL126749 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.680nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.690nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132072(3-(4-Formyl-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  0.730nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132067(CHEMBL129465 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  0.740nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132053(3-(2-Iodo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  0.75nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM3096(2-aminopyrido[2,3-d]pyrimidin-7(8H)-one deriv. | 6...)
Affinity DataKi:  0.800nMAssay Description:Displacement of (6-FAM)KI(pY)VV from full length PKMYT1 (unknown origin) by fluorescence polarization immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM3096(2-aminopyrido[2,3-d]pyrimidin-7(8H)-one deriv. | 6...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of human full length PKMYT1 expressed in HEK293 cells using EFS (247 to 259 residues) as substrate after 1 hr by fluorescence polarization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL25236 | CHEMBL540612 | N-(4-(4-(2-methoxyphe...)
Affinity DataKi:  0.920nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132042(3-Benzo[1,3]dioxol-5-yl-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132078(4-Acetyl-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-yl...)
Affinity DataKi:  1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132022(Biphenyl-4-carboxylic acid [4-((4aS,10bS)-7-hydrox...)
Affinity DataKi:  1nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50098203(1-{4-[2-(1H-Imidazol-4-yl)-ethylsulfanyl]-phenyl}-...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of [125I]-iodoproxyfan binding to human histamine H3 receptor of CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132024(3-(3-Iodo-phenyl)-N-{4-[4-(2-methoxy-phenyl)-piper...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132081(3-(2,4-Dichloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  1.28nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132061(3-(3,4-Dichloro-phenyl)-N-{4-[4-(2-methoxy-phenyl)...)
Affinity DataKi:  1.31nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [125I]-iodoproxyfan from rat histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50131926(CHEMBL127400 | CHEMBL129022 | Isoquinoline-3-carbo...)
Affinity DataKi:  1.48nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132038(5-Phenyl-penta-2,4-dienoic acid {4-[4-(2-methoxy-p...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Homo sapiens (Human))
University Munster

Curated by ChEMBL
LigandPNGBDBM50499215(CHEMBL3735947)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]ifenprodil from Glun2B receptor (unknown origin) expressed in mouse L(tk-) cell membranes after 120 mins by scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132025(2-Oxo-2H-chromene-3-carboxylic acid {4-[4-(2-metho...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50551241(CHEMBL4746028)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-(+)-pentazocine from Sigma1 receptor in guinea pig cortex membranes incubated for 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM3096(2-aminopyrido[2,3-d]pyrimidin-7(8H)-one deriv. | 6...)
Affinity DataKi:  2nMAssay Description:Displacement of (6-FAM)KI(pY)VV from PKMYT1 kinase domain (unknown origin) by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM3096(2-aminopyrido[2,3-d]pyrimidin-7(8H)-one deriv. | 6...)
Affinity DataKi:  2nMAssay Description:Displacement of (6-FAM)KI(pY)VV from PKMYT1 kinase domain (unknown origin) by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM3096(2-aminopyrido[2,3-d]pyrimidin-7(8H)-one deriv. | 6...)
Affinity DataKi:  2nMAssay Description:Inhibition of N-[3',6'-dihydroxy-3-oxo-3H-spiro(2-benzofuran-1,9'-xanthen)-5-yl]-N'-[2-(4-{4-[N-(2-chloro-6-methylphenyl)-5-carboxamido]-thiazol-2-yl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50071197(4-(4-Phenyl-butyl)-1H-imidazole | CHEMBL296450)
Affinity DataKi:  2.10nMAssay Description:Inhibition of [125I]-iodoproxyfan binding to human histamine H3 receptor of CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Und Medizinische Chemie Der Universit£T M£Nster

Curated by ChEMBL
LigandPNGBDBM50551242(CHEMBL4740593)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DTG from sigma 2 receptor in rat liver membranes incubated for 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132041(CHEMBL129429 | N-{4-[4-(2-Methoxy-phenyl)-piperazi...)
Affinity DataKi:  2.14nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM4213(6-(2,6-dichlorophenyl)-8-methyl-2-{[4-(morpholin-4...)
Affinity DataKi:  2.30nMAssay Description:Displacement of (6-FAM)KI(pY)VV from full length PKMYT1 (unknown origin) by fluorescence polarization immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase(Homo sapiens (Human))
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM4213(6-(2,6-dichlorophenyl)-8-methyl-2-{[4-(morpholin-4...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human full length PKMYT1 expressed in HEK293 cells using EFS (247 to 259 residues) as substrate after 1 hr by fluorescence polarization...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  2.40nMAssay Description:Inhibition of [125I]-iodoproxyfan binding to human histamine H3 receptor of CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50132030(4-Benzoyl-N-{4-[4-(2-methoxy-phenyl)-piperazin-1-y...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]-iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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