Affinity DataKi: 4.80nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of human LDHA using sodium pyruvate as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Mixed inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubated for 10 m...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 5.46E+3nMAssay Description:Competitive inhibition of human LDH5 meaured for 3 mins in presence of pyruvate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.46E+3nMAssay Description:Inhibition of LDHA in human liver using pyruvate as substrate incubated for 3 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
Affinity DataKi: 6.50E+3nMAssay Description:Non-competitive inhibition of human LDHA assessed as reduction in lactate production using pyruvate as substrate in presence of NADH by Lineweaver-Bu...More data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of human LDHA using pyruvate as substrate assessed as disappearance of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of human LDH-A using pyruvate as substrate and NADH as cofactor at 125 uM after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nMAssay Description:Non-competitive inhibition of human LDHA assessed as reduction in lactate production using pyruvate as substrate in presence of NADH by Lineweaver-Bu...More data for this Ligand-Target Pair
Affinity DataKi: 8.90E+3nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 9.10E+3nMAssay Description:Competitive inhibition of human LDH5 in presence of NADHMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+4nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Non-competitive inhibition of human LDHA assessed as reduction in lactate production using pyruvate as substrate in presence of NADH by Lineweaver-Bu...More data for this Ligand-Target Pair
Affinity DataKi: 1.57E+4nMAssay Description:Competitive inhibition of human LDH-A using pyruvate as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+4nMAssay Description:Competitive inhibition of human LDH5 incubated for 15 mins in presence of NADH by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.98E+4nMAssay Description:Competitive inhibition of human LDH-A using NADH as substrate after 5 mins by calorimetric assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+4nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Non-competitive inhibition of human LDHA assessed as reduction in lactate production using pyruvate as substrate in presence of NADH by Lineweaver-Bu...More data for this Ligand-Target Pair