Affinity DataKd: 1.70nMAssay Description:Binding affinity to human PIM2 (1 to 291 residues) expressed in bacterial system by KINOMEScan assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.90nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 3.10nMAssay Description:Binding affinity to Pim-2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Average Binding Constant for PIM2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity to recombinant human full-length N-terminal GST-tagged PIM2 expressed in baculovirus expression system using S6K2 peptide as substra...More data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding affinity to human PIM2More data for this Ligand-Target Pair
Affinity DataIC50: 49nM Kd: 23nMAssay Description:In vitro biochemical assays were performed in parallel to determine the most potent tool compound.More data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Competitive binding affinity to PIM2 in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKd: 130nMAssay Description:Average Binding Constant for PIM2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to human PIM2More data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Binding affinity to PIM2More data for this Ligand-Target Pair
Affinity DataKd: 460nMAssay Description:Average Binding Constant for PIM2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 650nMAssay Description:Average Binding Constant for PIM2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 680nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 770nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 770nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 770nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 870nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMAssay Description:Binding affinity to human PIM2 assessed as displacement of immobilized ligand by KINOMEscan scanMAX assay relative to controlMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 3.10E+3nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.20E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
Affinity DataKd: 5.00E+3nMAssay Description:Average Binding Constant for PIM2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 6.50E+3nMAssay Description:HS38 was evaluated using a P-33 ATP filter-binding assay by the International Centre for Kinase Profiling (University of Dundee) against 124 purified...More data for this Ligand-Target Pair
Affinity DataKd: 7.40E+3nMAssay Description:Binding affinity to human PIM2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for PIM2 kinase domainMore data for this Ligand-Target Pair