Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 1514
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM328995(1137478-47-7 | US11787792, Compound Y-154 | US9663...)
Affinity DataIC50:  1nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM328993(5-[[4-[[(2R)-morpholin-2-yl]methylamino]-5-(triflu...)
Affinity DataIC50:  1.40nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM328996(1137477-07-6 | US11787792, Compound Y-081 | US9663...)
Affinity DataIC50:  2nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM328997(1137478-45-5 | US11787792, Compound Y-152 | US9663...)
Affinity DataIC50:  2nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM328998(1137478-52-4 | US11787792, Compound Y-158 | US9663...)
Affinity DataIC50:  2nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM328994(5-[[4-[[(2S)-morpholin-2-yl]methylamino]-5-(triflu...)
Affinity DataIC50:  2.10nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM328999(1137478-38-6 | US11787792, Compound Y-147 | US9663...)
Affinity DataIC50:  4nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329000(1137478-46-6 | US11787792, Compound Y-153 | US9663...)
Affinity DataIC50:  4nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329001(1137478-48-8 | US11787792, Compound Y-155 | US9663...)
Affinity DataIC50:  5nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329002(1137478-40-0 | US11787792, Compound Y-149 | US9663...)
Affinity DataIC50:  10nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329003(1137478-50-2 | US11787792, Compound Y-156 | US9663...)
Affinity DataIC50:  10nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329004(1168103-91-0 | US11787792, Compound Y-146 | US9663...)
Affinity DataIC50:  11nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329005(1137478-39-7 | US11787792, Compound Y-148 | US9663...)
Affinity DataIC50:  13nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329006(1137478-51-3 | US11787792, Compound Y-157 | US9663...)
Affinity DataIC50:  15nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329007(1137478-41-1 | US11787792, Compound Y-150 | US9663...)
Affinity DataIC50:  17nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329008(1137477-35-0 | US11787792, Compound Y-102 | US9663...)
Affinity DataIC50:  20nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329009(1137478-54-6 | US11787792, Compound Y-159 | US9663...)
Affinity DataIC50:  23nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM329010(1137478-44-4 | US11787792, Compound Y-151 | US9663...)
Affinity DataIC50:  24nMAssay Description:CHK1 kinase activity was measured in a microfluidic assay that monitors the separation of a phosphorylated product from its substrate. The assay was ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent