Compile Data Set for Download or QSAR
maximum 50k data
Found 95 Enz. Inhib. hit(s) with all data for entry = 50015570
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21367(6-{4-[2-(methylsulfanyl)phenyl]piperazin-1-yl}-N-(...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21392(3-(2-aminoethyl)-1H-indole-5-carboxamide | 5-CT | ...)
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21370(6-[4-(2-acetylphenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21370(6-[4-(2-acetylphenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  4.14nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157768(5-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-t...)
Affinity DataKi:  6.05nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21368(6-[4-(2-methoxyphenyl)piperazin-1-yl]-N-(1,2,3,4-t...)
Affinity DataKi:  6.64nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21368(6-[4-(2-methoxyphenyl)piperazin-1-yl]-N-(1,2,3,4-t...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157768(5-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-t...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21371(6-[4-(2-hydroxyphenyl)piperazin-1-yl]-N-(1,2,3,4-t...)
Affinity DataKi:  11.4nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21369(6-[4-(2-methylphenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  15.2nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21375(6-[4-(2-cyanophenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  16.6nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157777(CHEMBL390558 | N-(5-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157780(CHEMBL426723 | N-(6-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  23.2nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21371(6-[4-(2-hydroxyphenyl)piperazin-1-yl]-N-(1,2,3,4-t...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157777(CHEMBL390558 | N-(5-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  24.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157779(CHEMBL225252 | N-(5-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  28.2nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157781(CHEMBL449089 | N-(6-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157766(CHEMBL222262 | N-(8-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157766(CHEMBL222262 | N-(8-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  31.4nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157767(CHEMBL376662 | N-(5-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157787(CHEMBL376531 | N-(7-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  38.4nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157771(CHEMBL221732 | N-(7-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21374(6-[4-(2-chlorophenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  40.1nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157771(CHEMBL221732 | N-(7-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157780(CHEMBL426723 | N-(6-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  43.1nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21375(6-[4-(2-cyanophenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  48.7nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21367(6-{4-[2-(methylsulfanyl)phenyl]piperazin-1-yl}-N-(...)
Affinity DataKi:  52.7nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157779(CHEMBL225252 | N-(5-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  54.4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157781(CHEMBL449089 | N-(6-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21373(6-[4-(2-nitrophenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  63.3nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157782(CHEMBL225441 | N-(8-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21372(6-(4-phenylpiperazin-1-yl)-N-(1,2,3,4-tetrahydrona...)
Affinity DataKi:  65.6nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157784(4-(2,5-dimethoxyphenyl)-N-(1,2,3,4-tetrahydronapht...)
Affinity DataKi:  70.3nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157782(CHEMBL225441 | N-(8-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21372(6-(4-phenylpiperazin-1-yl)-N-(1,2,3,4-tetrahydrona...)
Affinity DataKi:  77.8nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Wistar Han rat cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157787(CHEMBL376531 | N-(7-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  78.9nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157770(4-(4-(2-methoxyphenyl)piperazin-1-yl)-N-(1,2,3,4-t...)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21374(6-[4-(2-chlorophenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157783(4-(3-cyanophenyl)-N-(1,2,3,4-tetrahydronaphthalen-...)
Affinity DataKi:  97.8nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157765(4-(3-methoxyphenyl)-N-(1,2,3,4-tetrahydronaphthale...)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157765(4-(3-methoxyphenyl)-N-(1,2,3,4-tetrahydronaphthale...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157769(4-(4-chloro-2-methoxyphenyl)-N-(1,2,3,4-tetrahydro...)
Affinity DataKi:  122nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157772(4-(1,2-benzisoxazol-3-yl)-N-(1,2,3,4-tetrahydronap...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21372(6-(4-phenylpiperazin-1-yl)-N-(1,2,3,4-tetrahydrona...)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157785(CHEMBL390062 | N-(7-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157765(4-(3-methoxyphenyl)-N-(1,2,3,4-tetrahydronaphthale...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Wistar Han rat cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157773(CHEMBL224929 | N-(8-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]LSD from rat recombinant 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50157785(CHEMBL390062 | N-(7-methoxy-1,2,3,4-tetrahydronaph...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM21373(6-[4-(2-nitrophenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  183nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in Wistar Han rat hippocampal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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