Compile Data Set for Download or QSAR
Report error Found 102 for UniProtKB: O08786
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50245192(3-((S)-4-(1-(3-ethoxyphenyl)-2-(2-fluoro-4-methylp...)
Affinity DataEC50:  0.0340nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50245205(2-((S)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50245186(3-((S)-4-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazol...)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50343722(3-(4-(5-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-4-(2...)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at mouse CCK1 receptor expressed in CHO Flip cells assessed as increase in radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50245189(3-((R)-3-(acetamidomethyl)-4-(1-(3-ethoxyphenyl)-2...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50016425(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataKi:  0.191nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.300nMAssay Description:Potency in displacing [3H]propionyl-Cholecystokinin from mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50245187(CHEMBL504861 | CHEMBL446789 | 3-(4-(1-(3-ethoxyphe...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.491nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50245195(2-(((R)-1-(1-(3-ethoxyphenyl)-2-p-tolyl-1H-imidazo...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50343721(3-(4-(4-(2-fluoro-4-methylphenyl)-5-(4-methoxyphen...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at mouse CCK1 receptor expressed in CHO Flip cells assessed as increase in radio labeled inositol phosphate accumulation by Wallac m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50245180(CHEMBL505409 | CHEMBL505727 | 3-(4-(1-(3-ethoxyphe...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at mouse CCK1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226755(CHEMBL415630)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50024317(Tetragastrin | CHEMBL120632 | 3-{2-[2-Amino-3-(1H-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50073050((S)-1-(3-Amino-pentanoyl)-2,3-dihydro-1H-indole-2-...)
Affinity DataKi:  7nMAssay Description:Binding affinity in Cholecystokinin type A receptor binding assay (iv) in miceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284146([(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 14nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284148([(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 46nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284156([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 64nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50016424(N-(2-Amino-1-benzyl-ethyl)-3-{2-[2-{[9-tert-butoxy...)
Affinity DataKi:  120nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287255(N-[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-ethy...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]pentagastrin from Cholecystokinin receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287234(3-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287253(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284147([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 270nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50016426(3-{2-[2-(6-Amino-2-{2-[2-(2-tert-butoxycarbonylami...)
Affinity DataKi:  300nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287265({2-[3-(3-Piperidin-1-ylmethyl-phenoxy)-propylcarba...)
Affinity DataIC50: 310nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287250(4-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50: 330nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287251(N-[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-ethy...)
Affinity DataIC50: 330nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287256(6-(2-{3-[3-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50: 340nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287233(N-[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-ethy...)
Affinity DataIC50: 380nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287259(N-[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-ethy...)
Affinity DataIC50: 390nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287244(2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihydro...)
Affinity DataIC50: 430nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284160([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 430nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284161((E)-N-[(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine...)
Affinity DataIC50: 520nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287248(N-[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-ethy...)
Affinity DataIC50: 560nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284151(((2S,5S)-1-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-...)
Affinity DataIC50: 630nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287238(6-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50: 650nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287236(N-[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-ethy...)
Affinity DataIC50: 720nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287272([2-(4-{2-[3-(3-Piperidin-1-ylmethyl-phenoxy)-propy...)
Affinity DataIC50: 740nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287254(N-{[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-eth...)
Affinity DataIC50: 760nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284158(((2S,5S)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 840nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287246(4-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50: 900nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50016421(3-{2-[2-(6-Amino-2-{2-[2-(2-tert-butoxycarbonylami...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity measured by inhibiting [3H]Boc[Nle28,31]CCK27-33 specific binding to Cholecystokinin receptor in mouse brain membranes at a KD conce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287271((3-{2-[2-(2,2-Diamino-vinyl)-thiazol-4-ylmethylsul...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287239(N-{[2-(2-Guanidino-thiazol-4-ylmethylsulfanyl)-eth...)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287261((3-{2-[2-(2,2-Diamino-vinyl)-thiazol-4-ylmethylsul...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50287252(3-{2-[2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3-dihy...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against Cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
Merck

Curated by ChEMBL
LigandPNGBDBM50284159(((2S,5S)-5-Benzyl-1-{(S)-2-[(1H-indole-3-carbonyl)...)
Affinity DataIC50: 1.40E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

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