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TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014738(CHEMBL130253 | N-(Adamantyl-sulfonyl)-N-(methoxy s...)
Affinity DataKi:  15nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014747(CHEMBL131780 | 3-[(1-{2-[(1-Acetyl-pyrrolidine-2-c...)
Affinity DataKi:  29nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50312532(molassamide | CHEMBL1077010)
Affinity DataIC50: 32nMAssay Description:Inhibition of pig pancreatic elastase preincubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014736(CHEMBL337396 | (1-{1-Methyl-2-oxo-2-[2-(3,3,3-trif...)
Affinity DataKi:  32nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014730(CHEMBL130271 | N-(1-{1-Methyl-2-oxo-2-[2-(3,3,3-tr...)
Affinity DataKi:  33nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071966((R)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071973((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071968((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014732(CHEMBL339870 | 1-{2-[2-(5-Dimethylamino-naphthalen...)
Affinity DataKi:  88nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014745(CHEMBL131188 | 3-{2-[2-(2-Benzyloxycarbonylamino-p...)
Affinity DataKi:  140nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014742(CHEMBL130128 | Acetyl-Ala-Ala-Pro-Ala-triflurometh...)
Affinity DataKi:  150nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071983(CHEMBL310738 | (S)-3-((S)-2-Acetylamino-3-carboxy-...)
Affinity DataIC50: 190nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014740(CHEMBL130718 | Acetyl-Pro-Ala-Pro-Ala-trifluoro me...)
Affinity DataKi:  240nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50015856(CHEMBL313754 | 3-Acetoxymethyl-7-formyloxy-5,5,8-t...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014748(CHEMBL436383 | 3-[(1-{2-[2-(3-Methoxycarbonyl-prop...)
Affinity DataKi:  680nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014744(CHEMBL335981 | 3-[(1-{2-[(1-Acetyl-pyrrolidine-2-c...)
Affinity DataKi:  690nMAssay Description:Binding affinity against porcine pancreatic ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50228470(CHEMBL2370693)
Affinity DataKi:  800nMAssay Description:Binding affinity against porcine pancreatic ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014737(CHEMBL446422 | {1-Benzyl-2-oxo-2-[2-(3,3,3-trifluo...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50015876(CHEMBL84768 | 7-Acetoxy-3-acetoxymethyl-5,5,8-trio...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071965((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 2.20E+3nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226399(CHEMBL3143932)
Affinity DataKi:  2.40E+3nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50429202(LYNGBYASTATIN 7)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50479189(CHEBI:66142 | KEMPOPEPTIN A)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50479190(SOMAMIDE B)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405198(CHEMBL52356)
Affinity DataKi:  8.13E+3nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014733(CHEMBL340062 | 2,2-Difluoro-4-[(1-{2-[2-(3-methoxy...)
Affinity DataKi:  9.90E+3nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50302107(Grassystatin A | CHEMBL567893)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine pancreatic elastase after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405207(CHEMBL53936)
Affinity DataKi:  1.51E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226400(CHEMBL3143923)
Affinity DataKi:  1.95E+4nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237204(Esculin laurate)
Affinity DataIC50: 2.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50015857(CHEMBL421718 | 3-Acetoxymethyl-5,5,8-trioxo-7-phen...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of Porcine pancreatic elastase (PPE) enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405196(CHEMBL54748)
Affinity DataKi:  2.14E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237205(Esculin myristate)
Affinity DataIC50: 2.50E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014734(CHEMBL132768 | N-{1-Benzyl-2-oxo-2-[2-(3,3,3-trifl...)
Affinity DataKi:  2.80E+4nMAssay Description:Binding affinity for porcine ElastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237206(Esculin palmitate)
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226396(CHEMBL3143922)
Affinity DataKi:  3.15E+4nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226401(CHEMBL3143927)
Affinity DataKi:  3.50E+4nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226397(CHEMBL3143925)
Affinity DataKi:  4.25E+4nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 5.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237207(Esculin stearate)
Affinity DataIC50: 6.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50479191(KEMPOPEPTIN B)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405203(CHEMBL54524)
Affinity DataKi:  6.92E+4nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50226398(CHEMBL3143926)
Affinity DataKi:  8.21E+4nMAssay Description:Compound is evaluated for the inhibition of porcine pancreatic (PP) elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237203(Esculin)
Affinity DataIC50: 1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237184(Rutin)
Affinity DataIC50: 1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237198(Phloridzin)
Affinity DataIC50: 1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405200(CHEMBL54583)
Affinity DataKi:  1.41E+5nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1/2A(Pig)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50071967((R)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)
Affinity DataIC50: 2.06E+5nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405194(CHEMBL50396)
Affinity DataKi:  2.51E+5nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50405202(CHEMBL52938)
Affinity DataKi:  3.16E+5nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PP elastase) expressed as inhibitory constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
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