Compile Data Set for Download or QSAR
Report error Found 244 of affinity data for UniProtKB/TrEMBL: Q9GZQ6
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50029188(CHEMBL2165920)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataKi:  0.0600nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402454(CHEMBL2208337)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50029188(CHEMBL2165920)
Affinity DataKi:  0.590nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583768(CHEMBL5093771)
Affinity DataKi:  0.730nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402459(CHEMBL2208301)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50565194(CHEMBL4793841)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-FFRF-NH2 from human NPFFR1 expressed in CHO cell membrane by Topcount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50037557(2-{[1-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-4...)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to human NPFFR1 expressed in green monkey COS-7 cell membranes by [125I]-1DMeNPFF radioligand based saturation binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50029188(CHEMBL2165920)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM86143(RFamide-related peptide 3 | L-Val-L-Pro-L-Asn-L-Le...)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human NPFF1 receptor expressed in COS1 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336911((S)-2-((S)-2-((S)-5-amino-2-((S)-1-((S)-2-((S)-2-(...)
Affinity DataIC50: 1.90nMAssay Description:Displacement of (D-[125I]Tyr1, MePhe3)-NPFF from NPFFR1 after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402449(CHEMBL2208325)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402453(CHEMBL2208338)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50037567(2-[(Pyrrolidine-2-carbonyl)-amino]-pentanedioic ac...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50565182(CHEMBL4797394)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]-1-DMe-NPFF from human NPFF1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50565178(CHEMBL4460742)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cells by gamma-counter methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50029188(CHEMBL2165920)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50029138(CHEMBL3360830)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50029138(CHEMBL3360830)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]YVP from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2016
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583765(CHEMBL5090293)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataIC50: 4.70nMAssay Description:Displacement of (D-[125I]Tyr1, MePhe3)-NPFF from NPFFR1 after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583777(CHEMBL5085324)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402452(CHEMBL2208320)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402451(CHEMBL2208322)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583770(CHEMBL5071745)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583767(CHEMBL5075638)
Affinity DataKi:  6.60nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402442(CHEMBL2208303)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583766(CHEMBL5074999)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50037567(2-[(Pyrrolidine-2-carbonyl)-amino]-pentanedioic ac...)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]-1DMeNPFF from human NPFFR1 expressed in HEK293 cells incubated for 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583769(CHEMBL5082175)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402444(CHEMBL2208319)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402457(CHEMBL2208340)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583773(CHEMBL5091013)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50442584(CHEMBL2440929)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]YVP from human NPFFR1 expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50060728((R)-5-(diaminomethyleneamino)-2-(2,2-diphenylaceta...)
Affinity DataKi:  12nMAssay Description:Binding affinity to human NPFF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50565185(CHEMBL4777535)
Affinity DataKi:  13nMAssay Description:Binding affinity to human NPFFR1 by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402443(CHEMBL2208299)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583775(CHEMBL5088703)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50555150(CHEMBL4793250)
Affinity DataEC50:  17nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50060728((R)-5-(diaminomethyleneamino)-2-(2,2-diphenylaceta...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]NPVF from human NPFF1 expressed in CHO cells by radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50555150(CHEMBL4793250)
Affinity DataEC50:  18nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50060728((R)-5-(diaminomethyleneamino)-2-(2,2-diphenylaceta...)
Affinity DataKd:  20.9nMAssay Description:Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50565180(CHEMBL4776204)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human NPFFR1 expressed in CHO-K1 cells assessed as reversal of agonist-induced inhibition of forskolin-stimulated cAMP accumul...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50583771(CHEMBL5084208)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]-1DMeNPFF from recombinant human NPFF1 receptor expressed in CHO cells by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
University of Strasbourg

Curated by ChEMBL
LigandPNGBDBM50402458(CHEMBL2208339)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]FFRF-NH2 from human flag-tagged NPFF1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Displayed 1 to 50 (of 244 total ) | Next | Last >>
Jump to: