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Compound Name:

Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
1 Ki 76 IC50
  • 3-phosphoinositide dependent protein kinase-1
  • ALK tyrosine kinase receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BDNF/NT-3 growth factors receptor
  • CDC7 and DBF4
  • Cyclin-Dependent Kinase 2 (CDK2)
  • Dual specificity protein kinase TTK
  • Epidermal growth factor receptor
  • Eukaryotic elongation factor 2 kinase
  • Fibroblast growth factor receptor 1
  • Focal adhesion kinase 1
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin receptor
  • Insulin-like growth factor I receptor
  • MAP kinase-activated protein kinase 2
  • Mast/stem cell growth factor receptor Kit
  • Maternal embryonic leucine zipper kinase
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 14
  • NT-3 growth factor receptor
  • PKC alpha and beta-2
  • Pancreatic endoplasmic reticulum kinase (PERK)
  • Platelet-derived growth factor receptor beta
  • Proto-oncogene tyrosine-protein kinase ROS
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase LMTK3
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase NIM1
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase pim-1
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 3
  • cAMP-dependent protein kinase (PKA)
  • US10081622, Compound 11
  • US10370379, Entrectinib
  • US9029356, 11
  • US9255087, 11
  • US9616059, 11
47 Ki 25 IC50 5 Kd
  • Benzodiazepine receptors; peripheral & central
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • Gamma-aminobutyric acid type B receptor subunit 1
  • Nuclear receptor subfamily 1 group I member 3
  • Peripheral-Type Benzodiazepine Receptor
  • Translocator protein
  • 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoquinoline-3-carboxamide
  • CHEMBL15313
  • N-(butan-2-yl)-1-(2-chlorophenyl)-N-methylisoquinoline-3-carboxamide
  • PK 11195
  • PK-11195
  • PK11195
  • RP 52028
  • [3H]PK 11195
74 IC50 3 Kd
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 3A
  • Activin receptor-like kinase 2 (ALK-2)(aa 172-499)
  • Adenosine receptor A1
  • Alpha-1A adrenergic receptor
  • Aurora kinase A/Targeting protein for Xklp2
  • Axin-1/Glycogen synthase kinase-3 beta
  • Bile salt export pump (BSEP)
  • D(1A) dopamine receptor
  • DNA (cytosine-5)-methyltransferase 1 (DNMT1)
  • EZH1/PRC2
  • EZH2/SUZ12/EED/RBBP7/RBBP4
  • Estrogen receptor
  • Fibroblast growth factor receptor 2 (FGFR2)
  • Fibroblast growth factor receptor 4 (FGFR4)
  • Gamma-aminobutyric acid receptor subunit alpha-1
  • Histone-arginine methyltransferase CARM1
  • Histone-lysine N-methyltransferase SETDB1
  • Histone-lysine N-methyltransferase SMYD3
  • Histone-lysine N-methyltransferase SUV39H2 (Suv39H2)
  • Histone-lysine N-methyltransferase, H3 lysine-79 specific
  • Interleukin-1 receptor-associated kinase 1 (IRAK1)
  • Interleukin-1 receptor-associated kinase 4
  • Kinase insert domain receptor (KDR)
  • MLL
  • Mitogen-activated protein kinase kinase kinase 8 (MAP3K8)
  • Mitogen-activated protein kinase kinase kinase kinase 4
  • Muscarinic acetylcholine receptor M2
  • N-lysine methyltransferase SETD6 (SETD6)
  • Nuclear SET domain-containing protein 1 (NSD1)
  • Nuclear SET domain-containing protein 2 (NSD2)
  • Nuclear SET domain-containing protein 3 (NSD3)
  • Nuclear receptor subfamily 1 group I member 2
  • PRMT5/MEP50 Enzyme
  • Platelet-derived growth factor receptor alpha (PDGFRa)
  • Polycomb protein EED (EED)
  • Polycomb repressive complex 2 (PRC2)
  • Potassium voltage-gated channel subfamily H member 2
  • Protein G9a (G9a)
  • Protein arginine methyltransferase 3 (PRMT3)
  • Protein arginine methyltransferase 8 (PRMT8)
  • Protein kinase C alpha type
  • Protein kinase C theta type
  • Protein-arginine N-methyltransferase 1
  • Receptor-type tyrosine-protein kinase FLT3 (FLT3)
  • Rho-associated protein kinase 2 (ROCK2)
  • SET and MYND domain-containing protein 2 (SMYD2)
  • SET domain-containing protein 2 (SETD2)
  • SET domain-containing protein 7/9 (Set7/9)
  • SET domain-containing protein 8 (SetD8)
  • Serine/threonine-protein kinase 17B (STK17B)
  • Serine/threonine-protein kinase 4 (STK4)
  • Sodium-dependent dopamine transporter
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase ZAP-70
  • alpha-1 Nicotinic AChR
  • EED226
74 IC50 3 Kd
  • Cereblon/Histone deacetylase 1
  • Cereblon/Histone deacetylase 2
  • Cereblon/Histone deacetylase 4
  • Cereblon/Histone deacetylase 6
  • Histone deacetylase 1
  • Histone deacetylase 10
  • Histone deacetylase 11
  • Histone deacetylase 2
  • Histone deacetylase 3
  • Histone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)
  • Histone deacetylase 4
  • Histone deacetylase 5
  • Histone deacetylase 7
  • Histone deacetylase 8
  • Histone deacetylase 9
  • CHEMBL2170177
  • US10188756, Compound CN110