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19 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
7
Interaction kinetics of liposome-incorporated unsaturated fatty acids with fatty acid-binding protein 3 by surface plasmon resonance.EBI
Osaka University
2
Detection of Rap1A as a yessotoxin binding protein from blood cell membranes.EBI
Osaka University
5
Interaction of ladder-shaped polyethers with transmembrane alpha-helix of glycophorin A as evidenced by saturation transfer difference NMR and surface plasmon resonance.EBI
Osaka University
5
Prenylcoumarin with Rev-export inhibitory activity from Cnidii Monnieris Fructus.EBI
Osaka University
7
Surface plasmon resonance-based detection of ladder-shaped polyethers by inhibition detection method.EBI
Osaka University
34
G9a/GLP Modulators: Inhibitors to Degraders.EBI
Osaka University
8
Structural optimization of a lysine demethylase 5 inhibitor for improvement of its cellular activity.EBI
Osaka University
6
Discovery of Selective Histone Deacetylase 1 and 2 Inhibitors: Screening of a Focused Library Constructed by Click Chemistry, Kinetic Binding Analysis, and Biological Evaluation.EBI
Osaka University
25
Evolution of Slow-Binding Inhibitors Targeting Histone Deacetylase Isoforms.EBI
Osaka University
2
Synthetic RNA Modulators in Drug Discovery.EBI
Osaka University
5
Design, Synthesis, and Monoamine Oxidase B Selective Inhibitory Activity of EBI
Osaka University
5
Design, Synthesis, and Monoamine Oxidase Inhibitory Activity of (+)-Cinchonaminone and Its Simplified Derivatives.EBI
Osaka University
32
Structure-Activity Relationships of Pentacyclic Triterpenoids as Inhibitors of Cyclooxygenase and Lipoxygenase Enzymes.EBI
Osaka University
10
Correlation of indoleamine-2,3-dioxigenase 1 inhibitory activity of 4,6-disubstituted indazole derivatives and their heme binding affinity.EBI
Osaka University
4
Peptidomimetic modification improves cell permeation of bivalent farnesyltransferase inhibitors.EBI
Osaka University
18
A selective human H(4)-receptor agonist: (-)-2-cyano-1-methyl-3-[(2R,5R)-5- [1H-imidazol-4(5)-yl]tetrahydrofuran-2-y] methylguanidine.EBI
Osaka University
4
Semisynthesis and biological evaluation of a cotylenin A mimic derived from fusicoccin A.EBI
Osaka University
1
Stable C-N axial chirality in 1-aryluracil scaffold and differences in in vitro metabolic clearance between atropisomers of PDE4 inhibitor.EBI
Osaka University
6
Rational identification of natural organic compounds to target the intermolecular interaction between Foxm and DNA in colorectal cancer.BDB
Linyi People'S Hospital