BDBM181010 US9133197, 1
SMILES Cn1c(nc2c(N)nc(CCCCO)nc12)-n1nccn1
InChI Key InChIKey=LXKQSSJIYWOEPP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 181010
Affinity DataKi: 51nM ΔG°: -9.94kcal/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Sigma-Tau Industrie Farmaceutiche Riunite
US Patent
Affinity DataKi: 53nMpH: 7.4Assay Description:The protein concentration of membrane suspension was determined using the Bradford method (Pierce, Rockford, Ill., USA) with bovine albumin as standa...More data for this Ligand-Target Pair