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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM181010'
TargetAdenosine receptor A1(Homo sapiens (Human))
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181010(US9133197, 1)
Affinity DataKi:  51nM ΔG°:  -41.6kJ/molepH: 7.4 T: 2°CAssay Description:Competition binding experiments have been performed incubating membranes from CHO-K1 cells stably transfected with the human adenosine A1 receptor (c...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Sigma-Tau Industrie Farmaceutiche Riunite

US Patent
LigandPNGBDBM181010(US9133197, 1)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO-K1 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed