BDBM50081174 CHEMBL3421968

SMILES COc1cc(ccc1Nc1nccc(n1)-c1cn(C)c2cnccc12)N1CCN(C)CC1

InChI Key InChIKey=ZYVXTMKTGDARKR-UHFFFAOYSA-N

Data  2 KI  25 IC50  3 Kd

PDB links: 2 PDB IDs match this monomer.

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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50081174   

LigandPNGBDBM50081174(CHEMBL3421968)
Affinity DataIC50:  764nMAssay Description:Inhibition of recombinant human DYRK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scint...More data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50081174(CHEMBL3421968)
Affinity DataIC50:  1.90E+5nMAssay Description:Inhibition of Dyrk2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed