BDBM101530 US8530494, 29::US8530494, 7::US8530652, 57

SMILES CN(C)C[C@@H](NC(=O)N1Cc2c(Nc3ncnc4n(C)cnc34)[nH]nc2C1(C)C)c1ccccc1

InChI Key InChIKey=FFZVTVDOHCMWOO-QGZVFWFLSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 101530   

TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Agouron Pharmaceuticals

US Patent
LigandPNGBDBM101530(US8530494, 29 | US8530494, 7 | US8530652, 57)
Affinity DataKi:  14nM EC50:  2.5nMAssay Description:The enzymatic activity of PAK4 KD was measured by its ability to catalyzed the transfer of a phosphate residue from a nucleoside triphosphate to an a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Agouron Pharmaceuticals

US Patent
LigandPNGBDBM101530(US8530494, 29 | US8530494, 7 | US8530652, 57)
Affinity DataKi:  940nMAssay Description:The enzymatic activity of PAK4 KD was measured by its ability to catalyzed the transfer of a phosphate residue from a nucleoside triphosphate to an a...More data for this Ligand-Target Pair
In DepthDetails US Patent