BDBM342172 6-(4-fluorophenyl)-4-[4-[5-(4- fluorophenyl)-4H-1,2,4-triazol-3-yl]-1- piperidyl]-7H-pyrrolo[2,3-d]pyrimidine::US9771369, Compound P-3206
SMILES Fc1ccc(cc1)-c1cc2c(ncnc2[nH]1)N1CCC(CC1)c1nnc([nH]1)-c1ccc(F)cc1
InChI Key InChIKey=QAEBJNSATRRFQQ-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 342172
Affinity DataKi: 500nMAssay Description:The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...More data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Assays for biochemical cell-based activity of c-kit kinase are known in the art, for example, as described in U.S. Pat. Nos. 7,498,342 and 7,846,941,...More data for this Ligand-Target Pair